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RSC Medicinal Chemistry|March 4, 2026
Harnessing oligonucleotide architecture for potent multivalent inhibition of human carbonic anhydrasesEslam M Abbass, Federico Ladu, Justine Mansot, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|March 8, 2019
Novel Re(I) tricarbonyl coordination compounds based on 2-pyridyl-1,2,3-triazole derivatives bearing a 4-amino-substituted benzenesulfonamide arm: synthesis, crystal structure, computational studies and inhibitory activity against carbonic anhydrase I, II, and IX isoforms†Yassine Aimene, Romain Eychenne, Sonia Mallet-Ladeira, et al.Chemistry, an Asian Journal|February 12, 2016
Solution and Solid-State Analysis of Binding of 13-Substituted Berberine Analogues to Human Telomeric G-quadruplexesMarta Ferraroni, Carla Bazzicalupi, Francesco Papi, et al.Bioorganic & Medicinal Chemistry|May 31, 2022
Chlorinated benzothiadiazines inhibit angiogenesis through suppression of VEGFR2 phosphorylationBader I Huwaimel, Sravan Jonnalagadda, Shirisha Jonnalagadda, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|December 3, 2019
Benzothiazole derivatives as anticancer agentsAli Irfan, Fozia Batool, Syeda Andleeb Zahra Naqvi, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|January 21, 2021
Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs - a joint docking/molecular dynamics studyAlessandro Bonardi, Alessio Nocentini, Sameh Mohamed Osman, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|December 13, 2021
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeaeSimone Giovannuzzi, Nader S Abutaleb, Chad S Hewitt, et al.Bioorganic Chemistry|March 18, 2020
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitorsDavide Moi, Alessio Nocentini, Alessandro Deplano, et al.ACS Medicinal Chemistry Letters|November 20, 2020
Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium Vibrio choleraeAlessandro Bonardi, Alessio Nocentini, Roberta Cadoni, et al.Journal of Medicinal Chemistry|August 14, 2024
Optimization of Ethoxzolamide Analogs with Improved Pharmacokinetic Properties for In Vivo Efficacy against Neisseria gonorrhoeaeMolly S Youse, Nader S Abutaleb, Alessio Nocentini, et al.Pageof 29