Showing results (11-20 of 34) with videos related to
Sort By:
Pageof 4
Journal of Medicinal Chemistry|July 22, 2005
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A3 adenosine receptor antagonistsPier Giovanni Baraldi, Mojgan Aghazadeh Tabrizi, Delia Preti, et al.Bioorganic & Medicinal Chemistry|December 14, 2007
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonistsMojgan Aghazadeh Tabrizi, Pier Giovanni Baraldi, Delia Preti, et al.Bioorganic & Medicinal Chemistry Letters|October 16, 2004
Synthesis, radiolabeling, and preliminary biological evaluation of [3H]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl)-piperazine, a potent antagonist radioligand for the P2X7 receptorRomeo Romagnoli, Pier Giovanni Baraldi, Maria Giovanna Pavani, et al.Bioorganic & Medicinal Chemistry|February 20, 2007
N(6)-[(hetero)aryl/(cyclo)alkyl-carbamoyl-methoxy-phenyl]-(2-chloro)-5'-N-ethylcarboxamido-adenosines: the first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptorPier Giovanni Baraldi, Delia Preti, Mojgan Aghazadeh Tabrizi, et al.Journal of Medicinal Chemistry|January 29, 2013
Design, synthesis, and pharmacological properties of new heteroarylpyridine/heteroarylpyrimidine derivatives as CB(2) cannabinoid receptor partial agonistsMojgan Aghazadeh Tabrizi, Pier Giovanni Baraldi, Giulia Saponaro, et al.European Journal of Medicinal Chemistry|July 5, 2015
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect studyRomeo Romagnoli, Pier Giovanni Baraldi, Carlota Lopez-Cara, et al.Bioorganic & Medicinal Chemistry Letters|June 5, 2004
[3H]-MRE 2029-F20, a selective antagonist radioligand for the human A2B adenosine receptorsPier Giovanni Baraldi, Mojgan Aghazadeh Tabrizi, Delia Preti, et al.Journal of Medicinal Chemistry|January 19, 2007
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]- 9H-purin-9-yl]-N-ethyl-beta-D-ribofuranuronamide derivatives as useful templates for the development of A2B adenosine receptor agonistsPier Giovanni Baraldi, Delia Preti, Mojgan Aghazadeh Tabrizi, et al.Mini Reviews in Medicinal Chemistry|June 23, 2007
Allosteric enhancers for A1 adenosine receptorPier Giovanni Baraldi, Maria Antonietta Iaconinoto, Allan R Moorman, et al.Journal of Medicinal Chemistry|June 29, 2012
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as selective CB(2) cannabinoid receptor ligands: structural investigations around a novel class of full agonistsPier Giovanni Baraldi, Giulia Saponaro, Allan R Moorman, et al.Pageof 4