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Investigative Ophthalmology & Visual Science|January 24, 2013
Broad-spectrum virucidal activity of (NVC-422) N,N-dichloro-2,2-dimethyltaurine against viral ocular pathogens in vitroAndreas Jekle, Suriani Abdul Rani, Chris Celeri, et al.Bioorganic & Medicinal Chemistry Letters|December 17, 2009
Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacyclesRémy C Lemoine, Ann C Petersen, Lina Setti, et al.Bioorganic & Medicinal Chemistry Letters|September 22, 2010
Evaluation of amide replacements in CCR5 antagonists as a means to increase intrinsic permeability. Part 2: SAR optimization and pharmacokinetic profile of a homologous azacyle seriesJutta Wanner, Lijing Chen, Rémy C Lemoine, et al.Bioorganic & Medicinal Chemistry Letters|February 9, 2010
Evaluation of a 3-amino-8-azabicyclo[3.2.1]octane replacement in the CCR5 antagonist maravirocRémy C Lemoine, Ann C Petersen, Lina Setti, et al.Acta Ophthalmologica|September 14, 2012
N-chlorotaurine and its analogues N,N-dichloro-2,2-dimethyltaurine and N-monochloro-2,2-dimethyltaurine are safe and effective bactericidal agents in ex vivo corneal infection modelsBarbara Teuchner, Christian Eitzinger, Matthias Lutz, et al.Bioorganic & Medicinal Chemistry Letters|February 24, 2010
Evaluation of a 4-aminopiperidine replacement in several series of CCR5 antagonistsRémy C Lemoine, Ann C Petersen, Lina Setti, et al.Antimicrobial Agents and Chemotherapy|December 5, 2012
NVC-422 inactivates Staphylococcus aureus toxinsAndreas Jekle, Jungjoo Yoon, Meghan Zuck, et al.The Journal of Biological Chemistry|December 23, 2008
CD4-anchoring HIV-1 fusion inhibitor with enhanced potency and in vivo stabilityChanghua Ji, Erhard Kopetzki, Andreas Jekle, et al.Bioorganic & Medicinal Chemistry Letters|May 12, 2010
Synthesis, SAR and evaluation of [1,4']-bipiperidinyl-4-yl-imidazolidin-2-one derivatives as novel CCR5 antagonistsDavid M Rotstein, Stephen D Gabriel, Nicole Manser, et al.Antiviral Research|April 17, 2017
Structure-activity relationship analysis of mitochondrial toxicity caused by antiviral ribonucleoside analogsZhinan Jin, April Kinkade, Ishani Behera, et al.Pageof 5