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Astrid Kaiser

Showing results (31-40 of 44) with videos related to

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Journal of Medicinal Chemistry|November 1, 2013
Aminothiazole-featured pirinixic acid derivatives as dual 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 inhibitors with improved potency and efficiency in vivoThomas Hanke, Friederike Dehm, Stefanie Liening, et al.
Journal of Medicinal Chemistry|June 8, 2018
Boosting Anti-Inflammatory Potency of Zafirlukast by Designed PolypharmacologySimone Schierle, Cathrin Flauaus, Pascal Heitel, et al.
Journal of Medicinal Chemistry|December 21, 2023
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, et al.
Journal of Medicinal Chemistry|July 28, 2017
Nonacidic Farnesoid X Receptor ModulatorsDaniel Flesch, Sun-Yee Cheung, Jurema Schmidt, et al.
ACS Medicinal Chemistry Letters|June 22, 2019
Computer-Aided Selective Optimization of Side Activities of TalinololKerstin Hiesinger, Jan S Kramer, Janosch Achenbach, et al.
Journal of Medicinal Chemistry|February 29, 2024
Development of Selective Pyrido[2,3-<i>d</i>]pyrimidin-7(8<i>H</i>)-one-Based Mammalian STE20-Like (MST3/4) Kinase InhibitorsMarcel Rak, Amelie Menge, Roberta Tesch, et al.
Biochemical Pharmacology|September 28, 2016
Characterization of the molecular mechanism of 5-lipoxygenase inhibition by 2-aminothiazolesSimon B M Kretschmer, Stefano Woltersdorf, Dominik Vogt, et al.
Journal of Medicinal Chemistry|June 11, 2026
First Structure-Activity-Relationship Study of Potent G2A AntagonistsVictor Hernandez-Olmos, Jan Heering, Felix F Lillich, et al.
Journal of Medicinal Chemistry|November 24, 2015
N-Benzylbenzamides: A Novel Merged Scaffold for Orally Available Dual Soluble Epoxide Hydrolase/Peroxisome Proliferator-Activated Receptor γ ModulatorsRené Blöcher, Christina Lamers, Sandra K Wittmann, et al.
Journal of Medicinal Chemistry|January 13, 2025
Identification of a Chemical Probe for BLT2 Activation by Scaffold HoppingVictor Hernandez-Olmos, Jan Heering, Niklas Ildefeld, et al.
Pageof 5

Showing results (31-40 of 44) with videos related to

Sort By:
Pageof 5
Journal of Medicinal Chemistry|November 1, 2013
Aminothiazole-featured pirinixic acid derivatives as dual 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 inhibitors with improved potency and efficiency in vivoThomas Hanke, Friederike Dehm, Stefanie Liening, et al.
Journal of Medicinal Chemistry|June 8, 2018
Boosting Anti-Inflammatory Potency of Zafirlukast by Designed PolypharmacologySimone Schierle, Cathrin Flauaus, Pascal Heitel, et al.
Journal of Medicinal Chemistry|December 21, 2023
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, et al.
Journal of Medicinal Chemistry|July 28, 2017
Nonacidic Farnesoid X Receptor ModulatorsDaniel Flesch, Sun-Yee Cheung, Jurema Schmidt, et al.
ACS Medicinal Chemistry Letters|June 22, 2019
Computer-Aided Selective Optimization of Side Activities of TalinololKerstin Hiesinger, Jan S Kramer, Janosch Achenbach, et al.
Journal of Medicinal Chemistry|February 29, 2024
Development of Selective Pyrido[2,3-<i>d</i>]pyrimidin-7(8<i>H</i>)-one-Based Mammalian STE20-Like (MST3/4) Kinase InhibitorsMarcel Rak, Amelie Menge, Roberta Tesch, et al.
Biochemical Pharmacology|September 28, 2016
Characterization of the molecular mechanism of 5-lipoxygenase inhibition by 2-aminothiazolesSimon B M Kretschmer, Stefano Woltersdorf, Dominik Vogt, et al.
Journal of Medicinal Chemistry|June 11, 2026
First Structure-Activity-Relationship Study of Potent G2A AntagonistsVictor Hernandez-Olmos, Jan Heering, Felix F Lillich, et al.
Journal of Medicinal Chemistry|November 24, 2015
N-Benzylbenzamides: A Novel Merged Scaffold for Orally Available Dual Soluble Epoxide Hydrolase/Peroxisome Proliferator-Activated Receptor γ ModulatorsRené Blöcher, Christina Lamers, Sandra K Wittmann, et al.
Journal of Medicinal Chemistry|January 13, 2025
Identification of a Chemical Probe for BLT2 Activation by Scaffold HoppingVictor Hernandez-Olmos, Jan Heering, Niklas Ildefeld, et al.
Pageof 5