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Journal of Medicinal Chemistry|April 5, 2014
Biased ligand modulation of seven transmembrane receptors (7TMRs): functional implications for drug discoveryCraig C Correll, Brian A McKittrick
Bioorganic & Medicinal Chemistry|February 9, 2005
Discovery of melanin-concentrating hormone receptor R1 antagonists using high-throughput synthesisJing Su, Brian A McKittrick, Haiqun Tang, et al.
Bioorganic & Medicinal Chemistry Letters|June 30, 2006
Modification of the clozapine structure by parallel synthesisJing Su, Haiqun Tang, Brian A McKittrick, et al.
Bioorganic & Medicinal Chemistry Letters|March 23, 2002
Sulfide analogues as potent and selective M(2) muscarinic receptor antagonistsYuguang Wang, Samuel Chackalamannil, Zhiyong Hu, et al.
Bioorganic & Medicinal Chemistry Letters|April 26, 2011
Synthesis and SAR study of tricyclic sulfones as γ-secretase inhibitors: C-6 and C-8 positionsJing Su, Haiqun Tang, Brian A McKittrick, et al.
Bioorganic & Medicinal Chemistry Letters|December 31, 2008
Spiro-piperidine azetidinones as potent TRPV1 antagonistsDong Xiao, Anandan Palani, Robert Aslanian, et al.
Bioorganic & Medicinal Chemistry Letters|October 15, 2013
Identification of 2-aminooxazole amides as acyl-CoA: diacylglycerol acyltransferase 1 (DGAT1) inhibitors through scaffold hopping strategyHyunjin M Kim, Michelle D Smith, Jae-Hun Kim, et al.
Bioorganic & Medicinal Chemistry|June 19, 2007
SAR study of bicyclo[4.1.0]heptanes as melanin-concentrating hormone receptor R1 antagonists: taming hERGJing Su, Brian A McKittrick, Haiqun Tang, et al.
Bioorganic & Medicinal Chemistry Letters|January 12, 2010
Discovery of new SCH 39166 analogs as potent and selective dopamine D1 receptor antagonistsLi Qiang, T K Sasikumar, Duane A Burnett, et al.
Bioorganic & Medicinal Chemistry Letters|July 3, 2007
Synthesis of novel bicyclo[4.1.0]heptane and bicyclo[3.1.0]hexane derivatives as melanin-concentrating hormone receptor R1 antagonistsJing Su, Haiqun Tang, Brian A McKittrick, et al.
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