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Expert Opinion on Drug Discovery
|
February 23, 2019
A bright future for fragment-based drug discovery: what does it hold?
Célien Jacquemard, Esther Kellenberger
Journal of Chemical Information and Modeling
|
April 14, 2020
LIT-PCBA: An Unbiased Data Set for Machine Learning and Virtual Screening
Viet-Khoa Tran-Nguyen, Célien Jacquemard, Didier Rognan
Bioinformatics (Oxford, England)
|
December 26, 2021
Comparing transmembrane protein structures with ATOLL
Célien Jacquemard, Guillaume Bret, Thomas Grutter, et al.
Journal of Cheminformatics
|
March 24, 2019
Binding mode information improves fragment docking
Célien Jacquemard, Malgorzata N Drwal, Jérémy Desaphy, et al.
Viruses
|
August 10, 2021
Modeling of CCR5 Recognition by HIV-1 gp120: How the Viral Protein Exploits the Conformational Plasticity of the Coreceptor
Célien Jacquemard, Florian Koensgen, Philippe Colin, et al.
Journal of Chemical Information and Modeling
|
May 29, 2024
Benchmarking AlphaFold-Generated Structures of Chemokine-Chemokine Receptor Complexes
Lauri Urvas, Luca Chiesa, Guillaume Bret, et al.
Journal of Chemical Information and Modeling
|
April 18, 2017
Do Fragments and Crystallization Additives Bind Similarly to Drug-like Ligands?
Malgorzata N Drwal, Célien Jacquemard, Carlos Perez, et al.
RSC Medicinal Chemistry
|
April 18, 2022
Comprehensive analysis of commercial fragment libraries
Julia Revillo Imbernon, Célien Jacquemard, Guillaume Bret, et al.
Journal of Medicinal Chemistry
|
June 16, 2018
Structural Insights on Fragment Binding Mode Conservation
Malgorzata N Drwal, Guillaume Bret, Carlos Perez, et al.
Molecules (Basel, Switzerland)
|
July 21, 2019
Local Interaction Density (LID), a Fast and Efficient Tool to Prioritize Docking Poses
Célien Jacquemard, Viet-Khoa Tran-Nguyen, Malgorzata N Drwal, et al.
Page
of 2
Search research articles
Search
Showing results (1-10 of 12) with videos related to
Sort By:
Page
of 2
Expert Opinion on Drug Discovery
|
February 23, 2019
A bright future for fragment-based drug discovery: what does it hold?
Célien Jacquemard, Esther Kellenberger
Journal of Chemical Information and Modeling
|
April 14, 2020
LIT-PCBA: An Unbiased Data Set for Machine Learning and Virtual Screening
Viet-Khoa Tran-Nguyen, Célien Jacquemard, Didier Rognan
Bioinformatics (Oxford, England)
|
December 26, 2021
Comparing transmembrane protein structures with ATOLL
Célien Jacquemard, Guillaume Bret, Thomas Grutter, et al.
Journal of Cheminformatics
|
March 24, 2019
Binding mode information improves fragment docking
Célien Jacquemard, Malgorzata N Drwal, Jérémy Desaphy, et al.
Viruses
|
August 10, 2021
Modeling of CCR5 Recognition by HIV-1 gp120: How the Viral Protein Exploits the Conformational Plasticity of the Coreceptor
Célien Jacquemard, Florian Koensgen, Philippe Colin, et al.
Journal of Chemical Information and Modeling
|
May 29, 2024
Benchmarking AlphaFold-Generated Structures of Chemokine-Chemokine Receptor Complexes
Lauri Urvas, Luca Chiesa, Guillaume Bret, et al.
Journal of Chemical Information and Modeling
|
April 18, 2017
Do Fragments and Crystallization Additives Bind Similarly to Drug-like Ligands?
Malgorzata N Drwal, Célien Jacquemard, Carlos Perez, et al.
RSC Medicinal Chemistry
|
April 18, 2022
Comprehensive analysis of commercial fragment libraries
Julia Revillo Imbernon, Célien Jacquemard, Guillaume Bret, et al.
Journal of Medicinal Chemistry
|
June 16, 2018
Structural Insights on Fragment Binding Mode Conservation
Malgorzata N Drwal, Guillaume Bret, Carlos Perez, et al.
Molecules (Basel, Switzerland)
|
July 21, 2019
Local Interaction Density (LID), a Fast and Efficient Tool to Prioritize Docking Poses
Célien Jacquemard, Viet-Khoa Tran-Nguyen, Malgorzata N Drwal, et al.
Page
of 2