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Chemmedchem
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September 16, 2020
The Quest for the Best Dual Orexin Receptor Antagonist (Daridorexant) for the Treatment of Insomnia Disorders
Christoph Boss, John Gatfield, Christine Brotschi, et al.
Journal of Medicinal Chemistry
|
February 13, 2024
Discovery of a Novel Orally Active, Selective LPA Receptor Type 1 Antagonist, 4-(4-(2-Isopropylphenyl)-4-((2-methoxy-4-methylphenyl)carbamoyl)piperidin-1-yl)-4-oxobutanoic Acid, with a Distinct Molecular Scaffold
Cyrille Lescop, Christine Brotschi, Jodi T Williams, et al.
Chemmedchem
|
July 9, 2016
Discovery of Highly Potent Dual Orexin Receptor Antagonists via a Scaffold-Hopping Approach
Bibia Heidmann, John Gatfield, Catherine Roch, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 4, 2015
Substituted pyrrolidin-2-ones: Centrally acting orexin receptor antagonists promoting sleep. Part 2
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
Science Advances
|
March 1, 2024
A uniquely efficacious type of CFTR corrector with complementary mode of action
Valentina Marchesin, Lucile Monnier, Peter Blattmann, et al.
Chemmedchem
|
August 23, 2014
Structure-activity relationship, biological, and pharmacological characterization of the proline sulfonamide ACT-462206: a potent, brain-penetrant dual orexin 1/orexin 2 receptor antagonist
Christoph Boss, Catherine Roch-Brisbare, Michel A Steiner, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 23, 2014
Discovery of substituted lactams as novel dual orexin receptor antagonists. Synthesis, preliminary structure-activity relationship studies and efforts towards improved metabolic stability and pharmacokinetic properties. Part 1
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
March 12, 2025
The novel lysophosphatidic acid receptor 1-selective antagonist, ACT-1016-0707, has unique binding properties that translate into effective antifibrotic and anti-inflammatory activity in different models of pulmonary fibrosis
Magdalena Birker-Robaczewska, Maxime Boucher, Giulia Ranieri, et al.
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Search research articles
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Showing results (11-20 of 18) with videos related to
Sort By:
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This site can display upto 18 results.
Chemmedchem
|
September 16, 2020
The Quest for the Best Dual Orexin Receptor Antagonist (Daridorexant) for the Treatment of Insomnia Disorders
Christoph Boss, John Gatfield, Christine Brotschi, et al.
Journal of Medicinal Chemistry
|
February 13, 2024
Discovery of a Novel Orally Active, Selective LPA Receptor Type 1 Antagonist, 4-(4-(2-Isopropylphenyl)-4-((2-methoxy-4-methylphenyl)carbamoyl)piperidin-1-yl)-4-oxobutanoic Acid, with a Distinct Molecular Scaffold
Cyrille Lescop, Christine Brotschi, Jodi T Williams, et al.
Chemmedchem
|
July 9, 2016
Discovery of Highly Potent Dual Orexin Receptor Antagonists via a Scaffold-Hopping Approach
Bibia Heidmann, John Gatfield, Catherine Roch, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 4, 2015
Substituted pyrrolidin-2-ones: Centrally acting orexin receptor antagonists promoting sleep. Part 2
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
Science Advances
|
March 1, 2024
A uniquely efficacious type of CFTR corrector with complementary mode of action
Valentina Marchesin, Lucile Monnier, Peter Blattmann, et al.
Chemmedchem
|
August 23, 2014
Structure-activity relationship, biological, and pharmacological characterization of the proline sulfonamide ACT-462206: a potent, brain-penetrant dual orexin 1/orexin 2 receptor antagonist
Christoph Boss, Catherine Roch-Brisbare, Michel A Steiner, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 23, 2014
Discovery of substituted lactams as novel dual orexin receptor antagonists. Synthesis, preliminary structure-activity relationship studies and efforts towards improved metabolic stability and pharmacokinetic properties. Part 1
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
March 12, 2025
The novel lysophosphatidic acid receptor 1-selective antagonist, ACT-1016-0707, has unique binding properties that translate into effective antifibrotic and anti-inflammatory activity in different models of pulmonary fibrosis
Magdalena Birker-Robaczewska, Maxime Boucher, Giulia Ranieri, et al.
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of 2