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Journal of Medicinal Chemistry|March 17, 2018
Intrinsic Property Forecast Index (iPFI) as a Rule of Thumb for Medicinal Chemists to Remove a Phototoxicity LiabilityJean-François Fournier, Claire Bouix-Peter, Denis Duvert, et al.Bioorganic & Medicinal Chemistry Letters|February 2, 2024
Discovery of a novel series of selective macrocyclic PKCTheta inhibitorsStefano Crosignani, Sebastien Campos, Claire Bouix-Peter, et al.Beilstein Journal of Organic Chemistry|February 10, 2021
Novel library synthesis of 3,4-disubstituted pyridin-2(1<i>H</i>)-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperatureRomain Pierre, Anne Brethon, Sylvain A Jacques, et al.Molecular Therapy. Nucleic Acids|February 2, 2024
Multispecies-targeting siRNAs for the modulation of JAK1 in the skinQi Tang, Katherine Y Gross, Hassan H Fakih, et al.Bioorganic & Medicinal Chemistry Letters|May 1, 2018
Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acneEtienne Thoreau, Jean-Marie Arlabosse, Claire Bouix-Peter, et al.ACS Medicinal Chemistry Letters|November 22, 2019
Impact of Minor Structural Modifications on Properties of a Series of mTOR InhibitorsGilles Ouvry, Laurence Clary, Loïc Tomas, et al.Bioorganic & Medicinal Chemistry Letters|November 6, 2016
Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonistsGilles Ouvry, Claire Bouix-Peter, Fabrice Ciesielski, et al.Bioorganic & Medicinal Chemistry Letters|March 10, 2017
Identification of novel TACE inhibitors compatible with topical applicationGilles Ouvry, Yaël Berton, Yushma Bhurruth-Alcor, et al.Bioorganic & Medicinal Chemistry Letters|March 25, 2018
Sulfoximines as potent RORγ inverse agonistsGilles Ouvry, Franck Bihl, Claire Bouix-Peter, et al.Bioorganic & Medicinal Chemistry Letters|August 21, 2018
Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphomaJean-François Fournier, Yushma Bhurruth-Alcor, Branislav Musicki, et al.Pageof 2