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Bioorganic & Medicinal Chemistry Letters
|
June 29, 2010
Structure-activity relationships and in vivo activity of (1H-pyrazol-4-yl)acetamide antagonists of the P2X(7) receptor
Paul J Beswick, Andy Billinton, Laura J Chambers, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 20, 2010
Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
Laura J Chambers, Alexander J Stevens, Andrew P Moses, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 12, 2010
Identification of 2-oxo-N-(phenylmethyl)-4-imidazolidinecarboxamide antagonists of the P2X(7) receptor
Lee Abberley, Aude Bebius, Paul J Beswick, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 30, 2009
Second generation of BACE-1 inhibitors part 2: Optimisation of the non-prime side substituent
Nicolas Charrier, Brian Clarke, Emmanuel Demont, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 29, 2010
BACE-1 hydroxyethylamine inhibitors using novel edge-to-face interaction with Arg-296
Brian Clarke, Leanne Cutler, Emmanuel Demont, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 2, 2009
Second generation of BACE-1 inhibitors part 3: Towards non hydroxyethylamine transition state mimetics
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 12, 2009
Second generation of BACE-1 inhibitors. Part 1: The need for improved pharmacokinetics
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Journal of Medicinal Chemistry
|
May 7, 2008
Second generation of hydroxyethylamine BACE-1 inhibitors: optimizing potency and oral bioavailability
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 4, 2008
BACE-1 inhibitors part 1: identification of novel hydroxy ethylamines (HEAs)
Brian Clarke, Emmanuel Demont, Colin Dingwall, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 2, 2008
BACE-1 inhibitors part 2: identification of hydroxy ethylamines (HEAs) with reduced peptidic character
Brian Clarke, Emmanuel Demont, Colin Dingwall, et al.
Page
of 3
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Showing results (11-20 of 22) with videos related to
Sort By:
Page
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Bioorganic & Medicinal Chemistry Letters
|
June 29, 2010
Structure-activity relationships and in vivo activity of (1H-pyrazol-4-yl)acetamide antagonists of the P2X(7) receptor
Paul J Beswick, Andy Billinton, Laura J Chambers, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 20, 2010
Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
Laura J Chambers, Alexander J Stevens, Andrew P Moses, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 12, 2010
Identification of 2-oxo-N-(phenylmethyl)-4-imidazolidinecarboxamide antagonists of the P2X(7) receptor
Lee Abberley, Aude Bebius, Paul J Beswick, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 30, 2009
Second generation of BACE-1 inhibitors part 2: Optimisation of the non-prime side substituent
Nicolas Charrier, Brian Clarke, Emmanuel Demont, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 29, 2010
BACE-1 hydroxyethylamine inhibitors using novel edge-to-face interaction with Arg-296
Brian Clarke, Leanne Cutler, Emmanuel Demont, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 2, 2009
Second generation of BACE-1 inhibitors part 3: Towards non hydroxyethylamine transition state mimetics
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 12, 2009
Second generation of BACE-1 inhibitors. Part 1: The need for improved pharmacokinetics
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Journal of Medicinal Chemistry
|
May 7, 2008
Second generation of hydroxyethylamine BACE-1 inhibitors: optimizing potency and oral bioavailability
Nicolas Charrier, Brian Clarke, Leanne Cutler, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 4, 2008
BACE-1 inhibitors part 1: identification of novel hydroxy ethylamines (HEAs)
Brian Clarke, Emmanuel Demont, Colin Dingwall, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 2, 2008
BACE-1 inhibitors part 2: identification of hydroxy ethylamines (HEAs) with reduced peptidic character
Brian Clarke, Emmanuel Demont, Colin Dingwall, et al.
Page
of 3