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Journal of Medicinal Chemistry
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August 30, 2021
ω-Functionalized Lipid Prodrugs of HIV NtRTI Tenofovir with Enhanced Pharmacokinetic Properties
Nicole Pribut, Michael D'Erasmo, Madhuri Dasari, et al.
ACS Pharmacology & Translational Science
|
May 18, 2023
Discovery of 5'-Substituted 5-Fluoro-2'-deoxyuridine Monophosphate Analogs: A Novel Class of Thymidylate Synthase Inhibitors
Madhuri Dasari, Stephen C Pelly, Jiafeng Geng, et al.
ACS Medicinal Chemistry Letters
|
May 26, 2018
Discovery of <i>N</i>-Alkyl Piperazine Side Chain Based CXCR4 Antagonists with Improved Drug-like Properties
Yesim A Tahirovic, Valarie M Truax, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
January 20, 2018
Synthesis and SAR of 1,2,3,4-Tetrahydroisoquinoline-Based CXCR4 Antagonists
Robert J Wilson, Edgars Jecs, Eric J Miller, et al.
ACS Medicinal Chemistry Letters
|
February 20, 2018
Synthesis of Novel Tetrahydroisoquinoline CXCR4 Antagonists with Rigidified Side-Chains
Edgars Jecs, Eric J Miller, Robert J Wilson, et al.
Journal of Medicinal Chemistry
|
July 28, 2018
Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties
Huy H Nguyen, Michelle B Kim, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
May 19, 2016
Discovery of a Fluorinated Enigmol Analog with Enhanced in Vivo Pharmacokinetic and Anti-Tumor Properties
Eric J Miller, Suzanne G Mays, Mark T Baillie, et al.
ACS Medicinal Chemistry Letters
|
October 22, 2021
Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings
Huy H Nguyen, Yesim A Tahirovic, Valarie M Truax, et al.
ACS Pharmacology & Translational Science
|
September 19, 2025
Next-Generation Lipid Prodrugs Orally Deliver Tenofovir via Enhanced Chylomicron Incorporation
Hannah Beth Gold, Nicole Pribut, Esther L Outtrim, et al.
Journal of Medicinal Chemistry
|
April 6, 2026
Discovery of Novel 2-Morpholine Tetrahydroisoquinoline CXCR4 Antagonists with Unique Properties
Yesim Altas Tahirovic, Zafer Sahin, Edgars Jecs, et al.
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Search research articles
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Showing results (41-50 of 52) with videos related to
Sort By:
Page
of 6
Journal of Medicinal Chemistry
|
August 30, 2021
ω-Functionalized Lipid Prodrugs of HIV NtRTI Tenofovir with Enhanced Pharmacokinetic Properties
Nicole Pribut, Michael D'Erasmo, Madhuri Dasari, et al.
ACS Pharmacology & Translational Science
|
May 18, 2023
Discovery of 5'-Substituted 5-Fluoro-2'-deoxyuridine Monophosphate Analogs: A Novel Class of Thymidylate Synthase Inhibitors
Madhuri Dasari, Stephen C Pelly, Jiafeng Geng, et al.
ACS Medicinal Chemistry Letters
|
May 26, 2018
Discovery of <i>N</i>-Alkyl Piperazine Side Chain Based CXCR4 Antagonists with Improved Drug-like Properties
Yesim A Tahirovic, Valarie M Truax, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
January 20, 2018
Synthesis and SAR of 1,2,3,4-Tetrahydroisoquinoline-Based CXCR4 Antagonists
Robert J Wilson, Edgars Jecs, Eric J Miller, et al.
ACS Medicinal Chemistry Letters
|
February 20, 2018
Synthesis of Novel Tetrahydroisoquinoline CXCR4 Antagonists with Rigidified Side-Chains
Edgars Jecs, Eric J Miller, Robert J Wilson, et al.
Journal of Medicinal Chemistry
|
July 28, 2018
Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties
Huy H Nguyen, Michelle B Kim, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
May 19, 2016
Discovery of a Fluorinated Enigmol Analog with Enhanced in Vivo Pharmacokinetic and Anti-Tumor Properties
Eric J Miller, Suzanne G Mays, Mark T Baillie, et al.
ACS Medicinal Chemistry Letters
|
October 22, 2021
Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings
Huy H Nguyen, Yesim A Tahirovic, Valarie M Truax, et al.
ACS Pharmacology & Translational Science
|
September 19, 2025
Next-Generation Lipid Prodrugs Orally Deliver Tenofovir via Enhanced Chylomicron Incorporation
Hannah Beth Gold, Nicole Pribut, Esther L Outtrim, et al.
Journal of Medicinal Chemistry
|
April 6, 2026
Discovery of Novel 2-Morpholine Tetrahydroisoquinoline CXCR4 Antagonists with Unique Properties
Yesim Altas Tahirovic, Zafer Sahin, Edgars Jecs, et al.
Page
of 6