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Franco Lombardo

Showing results (11-20 of 36) with videos related to

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Journal of Medicinal Chemistry|July 17, 2009
In silico prediction of volume of distribution in human using linear and nonlinear models on a 669 compound data setGiuliano Berellini, Clayton Springer, Nigel J Waters, et al.
Journal of Medicinal Chemistry|February 20, 2004
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statisticsFranco Lombardo, R Scott Obach, Marina Y Shalaeva, et al.
Journal of Medicinal Chemistry|June 14, 2002
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding dataFranco Lombardo, R Scott Obach, Marina Y Shalaeva, et al.
Journal of Pharmaceutical Sciences|February 18, 2016
Systematic Evaluation of Wajima Superposition (Steady-State Concentration to Mean Residence Time) in the Estimation of Human Intravenous Pharmacokinetic ProfileFranco Lombardo, Giuliano Berellini, Laura R Labonte, et al.
Journal of Medicinal Chemistry|April 30, 2014
Clearance mechanism assignment and total clearance prediction in human based upon in silico modelsFranco Lombardo, R Scott Obach, Manthena V Varma, et al.
Molecular Pharmaceutics|August 13, 2024
Application of Mechanistic Multiparameter Optimization and Large-Scale <i>In Vitro</i> to <i>In Vivo</i> Pharmacokinetics Correlations to Small-Molecule Therapeutic ProjectsFabio Broccatelli, Vijayabhaskar Veeravalli, Daniel Cashion, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals|August 2, 2012
Oxidative ipso substitution of 2,4-difluoro-benzylphthalazines: identification of a rare stable quinone methide and subsequent GSH conjugateMithat Gunduz, Upendra A Argikar, Amin Kamel, et al.
Pharmaceutical Development and Technology|February 21, 2002
Stabilization of pharmaceuticals to oxidative degradationKenneth C Waterman, Roger C Adami, Karen M Alsante, et al.
Journal of Chemical Information and Modeling|June 9, 2015
Benefit of Retraining pKa Models Studied Using Internally Measured DataPeter Gedeck, Yipin Lu, Suzanne Skolnik, et al.
Journal of Medicinal Chemistry|June 14, 2017
In Silico Absorption, Distribution, Metabolism, Excretion, and Pharmacokinetics (ADME-PK): Utility and Best Practices. An Industry Perspective from the International Consortium for Innovation through Quality in Pharmaceutical DevelopmentFranco Lombardo, Prashant V Desai, Rieko Arimoto, et al.
Pageof 4

Showing results (11-20 of 36) with videos related to

Sort By:
Pageof 4
Journal of Medicinal Chemistry|July 17, 2009
In silico prediction of volume of distribution in human using linear and nonlinear models on a 669 compound data setGiuliano Berellini, Clayton Springer, Nigel J Waters, et al.
Journal of Medicinal Chemistry|February 20, 2004
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statisticsFranco Lombardo, R Scott Obach, Marina Y Shalaeva, et al.
Journal of Medicinal Chemistry|June 14, 2002
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding dataFranco Lombardo, R Scott Obach, Marina Y Shalaeva, et al.
Journal of Pharmaceutical Sciences|February 18, 2016
Systematic Evaluation of Wajima Superposition (Steady-State Concentration to Mean Residence Time) in the Estimation of Human Intravenous Pharmacokinetic ProfileFranco Lombardo, Giuliano Berellini, Laura R Labonte, et al.
Journal of Medicinal Chemistry|April 30, 2014
Clearance mechanism assignment and total clearance prediction in human based upon in silico modelsFranco Lombardo, R Scott Obach, Manthena V Varma, et al.
Molecular Pharmaceutics|August 13, 2024
Application of Mechanistic Multiparameter Optimization and Large-Scale <i>In Vitro</i> to <i>In Vivo</i> Pharmacokinetics Correlations to Small-Molecule Therapeutic ProjectsFabio Broccatelli, Vijayabhaskar Veeravalli, Daniel Cashion, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals|August 2, 2012
Oxidative ipso substitution of 2,4-difluoro-benzylphthalazines: identification of a rare stable quinone methide and subsequent GSH conjugateMithat Gunduz, Upendra A Argikar, Amin Kamel, et al.
Pharmaceutical Development and Technology|February 21, 2002
Stabilization of pharmaceuticals to oxidative degradationKenneth C Waterman, Roger C Adami, Karen M Alsante, et al.
Journal of Chemical Information and Modeling|June 9, 2015
Benefit of Retraining pKa Models Studied Using Internally Measured DataPeter Gedeck, Yipin Lu, Suzanne Skolnik, et al.
Journal of Medicinal Chemistry|June 14, 2017
In Silico Absorption, Distribution, Metabolism, Excretion, and Pharmacokinetics (ADME-PK): Utility and Best Practices. An Industry Perspective from the International Consortium for Innovation through Quality in Pharmaceutical DevelopmentFranco Lombardo, Prashant V Desai, Rieko Arimoto, et al.
Pageof 4