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EMBO Molecular Medicine
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April 7, 2026
Integrating chemical, genetic, and feasibility assessments for anti-tubercular target validation
Dirk Schnappinger, Steven J Berthel, Helena I M Boshoff, et al.
Journal of Medicinal Chemistry
|
August 14, 2025
Novel Inhibitors of <i>Plasmodium</i> Phosphatidylinositol 4-kinase IIIβ with Low Propensity for Resistance: Life Cycle Stage Activity and <i>In Vivo</i> Efficacy in a Humanized Mouse Malaria Infection Model
Godwin A Dziwornu, Mmakwena M Mmonwa, Dina Coertzen, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 20, 2015
Whole cell screen based identification of spiropiperidines with potent antitubercular properties
Subramanyam J Tantry, Giulia Degiacomi, Sreevalli Sharma, et al.
Journal of Medicinal Chemistry
|
August 20, 2021
1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in <i>Mycobacterium tuberculosis</i>
Lutete Peguy Khonde, Rudolf Müller, Grant A Boyle, et al.
Journal of Medicinal Chemistry
|
January 4, 2021
Antitubercular 2-Pyrazolylpyrimidinones: Structure-Activity Relationship and Mode-of-Action Studies
Candice Soares de Melo, Vinayak Singh, Alissa Myrick, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 11, 2014
Thiazolopyridone ureas as DNA gyrase B inhibitors: optimization of antitubercular activity and efficacy
Ramesh R Kale, Manoj G Kale, David Waterson, et al.
Journal of Medicinal Chemistry
|
October 4, 2013
Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B
Manoj G Kale, Anandkumar Raichurkar, Shahul Hameed P, et al.
Journal of Medicinal Chemistry
|
November 18, 2017
Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification Studies
Colin R Wilson, Richard K Gessner, Atica Moosa, et al.
Journal of Medicinal Chemistry
|
June 25, 2024
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of <i>Plasmodium falciparum</i> Phosphatidylinositol-4-kinase and Hemozoin Formation with <i>In Vivo</i> Efficacy
Godwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, et al.
Journal of Medicinal Chemistry
|
May 30, 2014
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity
Maruti Naik, Vaishali Humnabadkar, Subramanyam J Tantry, et al.
Page
of 36
Search research articles
Search
Showing results (341-350 of 351) with videos related to
Sort By:
Page
of 36
EMBO Molecular Medicine
|
April 7, 2026
Integrating chemical, genetic, and feasibility assessments for anti-tubercular target validation
Dirk Schnappinger, Steven J Berthel, Helena I M Boshoff, et al.
Journal of Medicinal Chemistry
|
August 14, 2025
Novel Inhibitors of <i>Plasmodium</i> Phosphatidylinositol 4-kinase IIIβ with Low Propensity for Resistance: Life Cycle Stage Activity and <i>In Vivo</i> Efficacy in a Humanized Mouse Malaria Infection Model
Godwin A Dziwornu, Mmakwena M Mmonwa, Dina Coertzen, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 20, 2015
Whole cell screen based identification of spiropiperidines with potent antitubercular properties
Subramanyam J Tantry, Giulia Degiacomi, Sreevalli Sharma, et al.
Journal of Medicinal Chemistry
|
August 20, 2021
1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in <i>Mycobacterium tuberculosis</i>
Lutete Peguy Khonde, Rudolf Müller, Grant A Boyle, et al.
Journal of Medicinal Chemistry
|
January 4, 2021
Antitubercular 2-Pyrazolylpyrimidinones: Structure-Activity Relationship and Mode-of-Action Studies
Candice Soares de Melo, Vinayak Singh, Alissa Myrick, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 11, 2014
Thiazolopyridone ureas as DNA gyrase B inhibitors: optimization of antitubercular activity and efficacy
Ramesh R Kale, Manoj G Kale, David Waterson, et al.
Journal of Medicinal Chemistry
|
October 4, 2013
Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B
Manoj G Kale, Anandkumar Raichurkar, Shahul Hameed P, et al.
Journal of Medicinal Chemistry
|
November 18, 2017
Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification Studies
Colin R Wilson, Richard K Gessner, Atica Moosa, et al.
Journal of Medicinal Chemistry
|
June 25, 2024
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of <i>Plasmodium falciparum</i> Phosphatidylinositol-4-kinase and Hemozoin Formation with <i>In Vivo</i> Efficacy
Godwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, et al.
Journal of Medicinal Chemistry
|
May 30, 2014
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity
Maruti Naik, Vaishali Humnabadkar, Subramanyam J Tantry, et al.
Page
of 36