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Drug Discovery Today
|
May 12, 2009
From fragment to clinical candidate--a historical perspective
Gianni Chessari, Andrew J Woodhead
Journal of Magnetic Resonance (San Diego, Calif. : 1997)
|
August 8, 2002
Resin dynamics contributes to the NMR line broadening of organic molecules grafted onto a polystyrene resin
Guy Lippens, Gianni Chessari, Jean-Michel Wieruszeski
Journal of Medicinal Chemistry
|
May 7, 2008
Recent developments in fragment-based drug discovery
Miles Congreve, Gianni Chessari, Dominic Tisi, et al.
Journal of Medicinal Chemistry
|
May 5, 2022
Electrostatic Complementarity in Structure-Based Drug Design
Benjamin D Cons, David G Twigg, Rajendra Kumar, et al.
Pharmacology Research & Perspectives
|
October 25, 2024
The preclinical pharmacokinetics of Tolinapant-A dual cIAP1/XIAP antagonist with in vivo efficacy
Vanessa Martins, George Ward, Tomoko Smyth, et al.
Nucleic Acids Research
|
February 22, 2003
Sequence-specific minor groove binding by bis-benzimidazoles: water molecules in ligand recognition
Christian Bailly, Gianni Chessari, Carolina Carrasco, et al.
Chemical Science
|
October 20, 2021
C-H functionalisation tolerant to polar groups could transform fragment-based drug discovery (FBDD)
Gianni Chessari, Rachel Grainger, Rhian S Holvey, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)
|
December 20, 2002
An evaluation of force-field treatments of aromatic interactions
Gianni Chessari, Christopher A Hunter, Caroline M R Low, et al.
ACS Central Science
|
May 30, 2023
Accelerated Chemical Reaction Optimization Using Multi-Task Learning
Connor J Taylor, Kobi C Felton, Daniel Wigh, et al.
Journal of Medicinal Chemistry
|
February 16, 2007
Diverse, high-quality test set for the validation of protein-ligand docking performance
Michael J Hartshorn, Marcel L Verdonk, Gianni Chessari, et al.
Page
of 4
Search research articles
Search
Showing results (1-10 of 33) with videos related to
Sort By:
Page
of 4
Drug Discovery Today
|
May 12, 2009
From fragment to clinical candidate--a historical perspective
Gianni Chessari, Andrew J Woodhead
Journal of Magnetic Resonance (San Diego, Calif. : 1997)
|
August 8, 2002
Resin dynamics contributes to the NMR line broadening of organic molecules grafted onto a polystyrene resin
Guy Lippens, Gianni Chessari, Jean-Michel Wieruszeski
Journal of Medicinal Chemistry
|
May 7, 2008
Recent developments in fragment-based drug discovery
Miles Congreve, Gianni Chessari, Dominic Tisi, et al.
Journal of Medicinal Chemistry
|
May 5, 2022
Electrostatic Complementarity in Structure-Based Drug Design
Benjamin D Cons, David G Twigg, Rajendra Kumar, et al.
Pharmacology Research & Perspectives
|
October 25, 2024
The preclinical pharmacokinetics of Tolinapant-A dual cIAP1/XIAP antagonist with in vivo efficacy
Vanessa Martins, George Ward, Tomoko Smyth, et al.
Nucleic Acids Research
|
February 22, 2003
Sequence-specific minor groove binding by bis-benzimidazoles: water molecules in ligand recognition
Christian Bailly, Gianni Chessari, Carolina Carrasco, et al.
Chemical Science
|
October 20, 2021
C-H functionalisation tolerant to polar groups could transform fragment-based drug discovery (FBDD)
Gianni Chessari, Rachel Grainger, Rhian S Holvey, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)
|
December 20, 2002
An evaluation of force-field treatments of aromatic interactions
Gianni Chessari, Christopher A Hunter, Caroline M R Low, et al.
ACS Central Science
|
May 30, 2023
Accelerated Chemical Reaction Optimization Using Multi-Task Learning
Connor J Taylor, Kobi C Felton, Daniel Wigh, et al.
Journal of Medicinal Chemistry
|
February 16, 2007
Diverse, high-quality test set for the validation of protein-ligand docking performance
Michael J Hartshorn, Marcel L Verdonk, Gianni Chessari, et al.
Page
of 4