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RSC Advances|May 13, 2022
One step access to oxindole-based β-lactams through Ugi four-center three-component reactionGiulia Rainoldi, Giordano Lesma, Claudia Picozzi, et al.
Journal of Combinatorial Chemistry|May 10, 2005
Combinatorial solid-phase synthesis of 6-hydroxy-1,2,3,4-tetrahydro-beta-carbolines from l-5-hydroxytryptophanBruno Danieli, Paola Giovanelli, Giordano Lesma, et al.
Organic Letters|August 17, 2002
Concise total synthesis of (+/-)-aloperine and 6-epi-aloperineDaniele Passarella, Marco Angoli, Alessandra Giardini, et al.
Combinatorial Chemistry & High Throughput Screening|November 15, 2006
Microwave-assisted, solid-phase synthesis of a chiral 1,2,3,4-tetrahydro-quinoline libraryGiordano Lesma, Bruno Danieli, Francesco Lodroni, et al.
The Journal of Organic Chemistry|February 3, 2016
Organocatalytic Asymmetric Biginelli-like Reaction Involving IsatinMattia Stucchi, Giordano Lesma, Fiorella Meneghetti, et al.
Beilstein Journal of Organic Chemistry|February 13, 2013
The diketopiperazine-fused tetrahydro-β-carboline scaffold as a model peptidomimetic with an unusual α-turn secondary structureFrancesco Airaghi, Andrea Fiorati, Giordano Lesma, et al.
Organic Letters|February 14, 2004
Total enantioselective synthesis of (-)-cytisineBruno Danieli, Giordano Lesma, Daniele Passarella, et al.
Organic & Biomolecular Chemistry|June 21, 2011
Addition of TMSCN to chiral ketimines derived from isatin. Synthesis of an oxindole-based peptidomimetic and a bioactive spirohydantoinAlessandro Sacchetti, Alessandra Silvani, Francesco G Gatti, et al.
The Journal of Organic Chemistry|November 25, 2003
Remote stereocenter discrimination in the enzymatic resolution of piperidine-2-ethanol. Short enantioselective synthesis of sedamine and allosedamineMarco Angoli, Alessio Barilli, Giordano Lesma, et al.
ACS Medicinal Chemistry Letters|August 20, 2015
Multicomponent Synthesis and Biological Evaluation of a Piperazine-Based Dopamine Receptor Ligand LibraryMattia Stucchi, Peter Gmeiner, Harald Huebner, et al.
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