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Bioconjugate Chemistry|July 31, 2023
Design of Highly Fluorinated Peptides for Cell-based <sup>19</sup>F NMRJiaqian Li, Steven E Kirberger, Yiao Wang, et al.ACS Medicinal Chemistry Letters|September 19, 2019
Systematically Mitigating the p38α Activity of Triazole-based BET InhibitorsAngela S Carlson, Huarui Cui, Anand Divakaran, et al.ACS Chemical Biology|November 3, 2020
Quantifying the Selectivity of Protein-Protein and Small Molecule Interactions with Fluorinated Tandem Bromodomain Reader ProteinsPrakriti Kalra, Logan McGraw, Jennifer R Kimbrough, et al.Angewandte Chemie (International Ed. in English)|September 25, 2020
Selective N-Terminal BET Bromodomain Inhibitors by Targeting Non-Conserved Residues and Structured Water Displacement*Huarui Cui, Anand Divakaran, Anil K Pandey, et al.Hepatology (Baltimore, Md.)|November 7, 2020
Endothelial p300 Promotes Portal Hypertension and Hepatic Fibrosis Through C-C Motif Chemokine Ligand 2-Mediated Angiocrine SignalingJinhang Gao, Bo Wei, Mengfei Liu, et al.Journal of Medicinal Chemistry|September 26, 2018
Molecular Basis for the N-Terminal Bromodomain-and-Extra-Terminal-Family Selectivity of a Dual Kinase-Bromodomain InhibitorAnand Divakaran, Siva K Talluri, Alex M Ayoub, et al.Journal of Medicinal Chemistry|July 8, 2021
4-Methyl-1,2,3-Triazoles as <i>N</i>-Acetyl-Lysine Mimics Afford Potent BET Bromodomain Inhibitors with Improved SelectivityHuarui Cui, Angela S Carlson, Mary A Schleiff, et al.European Journal of Medicinal Chemistry|March 10, 2023
From PROTAC to inhibitor: Structure-guided discovery of potent and orally bioavailable BET inhibitorsMladen Koravovic, Anand Mayasundari, Gordana Tasic, et al.Journal of Medicinal Chemistry|January 10, 2022
A Structure-based Design Approach for Generating High Affinity BRD4 D1-Selective Chemical ProbesHuarui Cui, Anand Divakaran, Zachariah J Hoell, et al.Nature Communications|July 28, 2021
Super enhancer regulation of cytokine-induced chemokine production in alcoholic hepatitisMengfei Liu, Sheng Cao, Li He, et al.Pageof 1