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Organic Letters|September 22, 2025
4-Nitrophenyl Sulfamates as Precursors Containing Acid-Labile Functional Groups for Sulfamidation with Weakly Nucleophilic AminesFumio Watanabe, Kazuo Hattori, Kihito Hada, et al.Bioorganic & Medicinal Chemistry Letters|October 26, 2013
The sulfamide moiety affords higher inhibitory activity and oral bioavailability to a series of coumarin dual selective RAF/MEK inhibitorsToshihiro Aoki, Ikumi Hyohdoh, Noriyuki Furuichi, et al.Journal of Medicinal Chemistry|December 10, 2016
Discovery of [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-(1H-indol-2-yl)methanone (CH5183284/Debio 1347), An Orally Available and Selective Fibroblast Growth Factor Receptor (FGFR) InhibitorHirosato Ebiike, Naoki Taka, Masayuki Matsushita, et al.ACS Medicinal Chemistry Letters|June 6, 2014
Optimizing the Physicochemical Properties of Raf/MEK Inhibitors by Nitrogen ScanningToshihiro Aoki, Ikumi Hyohdoh, Noriyuki Furuichi, et al.ACS Medicinal Chemistry Letters|June 6, 2014
Fluorine Scanning by Nonselective Fluorination: Enhancing Raf/MEK Inhibition while Keeping Physicochemical PropertiesIkumi Hyohdoh, Noriyuki Furuichi, Toshihiro Aoki, et al.Pageof 1