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Future Medicinal Chemistry
|
October 26, 2011
Is drug discovery dead?
John J Baldwin
Future Medicinal Chemistry
|
August 1, 2014
Pharmaceutical R&D: an age of change?
John J Baldwin
Future Medicinal Chemistry
|
June 11, 2015
Drug discovery and development 2014: Returning toward the norm?
John J Baldwin
Combinatorial Chemistry & High Throughput Screening
|
August 24, 2006
Exploring structure-activity relationships of tricyclic farnesyltransferase inhibitors using ECLiPS libraries
Laura L Rokosz, Chia-Yu Huang, John C Reader, et al.
Journal of Molecular Graphics & Modelling
|
August 16, 2014
An electronic environment and contact direction sensitive scoring function for predicting affinities of protein-ligand complexes in Contour(®)
Peter R Lindblom, Guosheng Wu, Zhijie Liu, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 6, 2005
Surfing the piperazine core of tricyclic farnesyltransferase inhibitors
Laura L Rokosz, Chia-Yu Huang, John C Reader, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 17, 2007
3,4-Diamino-2,5-thiadiazole-1-oxides as potent CXCR2/CXCR1 antagonists
Purakkattle Biju, Arthur Taveras, Younong Yu, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 18, 2005
Guiding farnesyltransferase inhibitors from an ECLiPS library to the catalytic zinc
Chia-Yu Huang, Tara M Stauffer, Corey L Strickland, et al.
Bioorganic & Medicinal Chemistry
|
December 27, 2005
Synthesis, biological evaluation, and pharmacokinetic study of prolyl-1-piperazinylacetic acid and prolyl-4-piperidinylacetic acid derivatives as VLA-4 antagonists
Jun Chiba, Gensuke Takayama, Tohru Takashi, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 8, 2004
Identified a morpholinyl-4-piperidinylacetic acid derivative as a potent oral active VLA-4 antagonist
Jun Chiba, Nobuo Machinaga, Tohru Takashi, et al.
Page
of 2
Search research articles
Search
Showing results (1-10 of 18) with videos related to
Sort By:
Page
of 2
Future Medicinal Chemistry
|
October 26, 2011
Is drug discovery dead?
John J Baldwin
Future Medicinal Chemistry
|
August 1, 2014
Pharmaceutical R&D: an age of change?
John J Baldwin
Future Medicinal Chemistry
|
June 11, 2015
Drug discovery and development 2014: Returning toward the norm?
John J Baldwin
Combinatorial Chemistry & High Throughput Screening
|
August 24, 2006
Exploring structure-activity relationships of tricyclic farnesyltransferase inhibitors using ECLiPS libraries
Laura L Rokosz, Chia-Yu Huang, John C Reader, et al.
Journal of Molecular Graphics & Modelling
|
August 16, 2014
An electronic environment and contact direction sensitive scoring function for predicting affinities of protein-ligand complexes in Contour(®)
Peter R Lindblom, Guosheng Wu, Zhijie Liu, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 6, 2005
Surfing the piperazine core of tricyclic farnesyltransferase inhibitors
Laura L Rokosz, Chia-Yu Huang, John C Reader, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 17, 2007
3,4-Diamino-2,5-thiadiazole-1-oxides as potent CXCR2/CXCR1 antagonists
Purakkattle Biju, Arthur Taveras, Younong Yu, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 18, 2005
Guiding farnesyltransferase inhibitors from an ECLiPS library to the catalytic zinc
Chia-Yu Huang, Tara M Stauffer, Corey L Strickland, et al.
Bioorganic & Medicinal Chemistry
|
December 27, 2005
Synthesis, biological evaluation, and pharmacokinetic study of prolyl-1-piperazinylacetic acid and prolyl-4-piperidinylacetic acid derivatives as VLA-4 antagonists
Jun Chiba, Gensuke Takayama, Tohru Takashi, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 8, 2004
Identified a morpholinyl-4-piperidinylacetic acid derivative as a potent oral active VLA-4 antagonist
Jun Chiba, Nobuo Machinaga, Tohru Takashi, et al.
Page
of 2