Showing results (1-10 of 14) with videos related to
Sort By:
Pageof 2
Journal of the American Chemical Society|November 14, 2017
Radical Multicomponent Carboamination of [1.1.1]PropellaneJunichiro Kanazawa, Katsuya Maeda, Masanobu UchiyamaInternational Journal of Oncology|January 19, 2008
Pyranicin, a non-classical annonaceous acetogenin, is a potent inhibitor of DNA polymerase, topoisomerase and human cancer cell growthShunya Takahashi, Yuko Yonezawa, Akemi Kubota, et al.ACS Medicinal Chemistry Letters|October 25, 2016
Concise SAR Exploration Based on the "Head-to-Tail" Approach: Discovery of PI4KIIIα Inhibitors Bearing Diverse ScaffoldsSatoru Noji, Noriyoshi Seki, Takaki Maeba, et al.European Journal of Medicinal Chemistry|September 25, 2018
Discovery of potent liver-selective stearoyl-CoA desaturase-1 (SCD1) inhibitors, thiazole-4-acetic acid derivatives, for the treatment of diabetes, hepatic steatosis, and obesityTetsuya Iida, Minoru Ubukata, Ikuo Mitani, et al.Scientific Reports|November 28, 2018
Ternary crystal structure of human RORγ ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interactionMasato Noguchi, Akihiro Nomura, Satoki Doi, et al.ACS Medicinal Chemistry Letters|May 31, 2021
Discovery of Selective Transforming Growth Factor β Type II Receptor Inhibitors as Antifibrosis AgentsShohei Miwa, Masahiro Yokota, Yoshifumi Ueyama, et al.Bioorganic & Medicinal Chemistry Letters|February 27, 2009
Novel N-substituted 2-phenyl-1-sulfonylamino-cyclopropane carboxylates as selective ADAMTS-5 (Aggrecanase-2) inhibitorsMakoto Shiozaki, Katsuya Maeda, Tomoya Miura, et al.Bioorganic & Medicinal Chemistry Letters|September 22, 2009
Synthesis and SAR of 2-phenyl-1-sulfonylaminocyclopropane carboxylates as ADAMTS-5 (Aggrecanase-2) inhibitorsMakoto Shiozaki, Hiroto Imai, Katsuya Maeda, et al.Journal of Medicinal Chemistry|June 9, 2020
Discovery of a Janus Kinase Inhibitor Bearing a Highly Three-Dimensional Spiro Scaffold: JTE-052 (Delgocitinib) as a New Dermatological Agent to Treat Inflammatory Skin DisordersSatoru Noji, Yoshinori Hara, Tomoya Miura, et al.Journal of Medicinal Chemistry|March 23, 2011
Discovery of (1S,2R,3R)-2,3-dimethyl-2-phenyl-1-sulfamidocyclopropanecarboxylates: novel and highly selective aggrecanase inhibitorsMakoto Shiozaki, Katsuya Maeda, Tomoya Miura, et al.Pageof 2