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Methods in Molecular Biology (Clifton, N.J.)|February 25, 2015
Protocol for fragment hoppingKevin B Teuscher, Haitao JiChemical Science|June 15, 2018
Direct α-heteroarylation of amides (α to nitrogen) and ethers through a benzaldehyde-mediated photoredox reactionYongqiang Zhang, Kevin B Teuscher, Haitao JiJournal of Medicinal Chemistry|December 10, 2016
A Versatile Method to Determine the Cellular Bioavailability of Small-Molecule InhibitorsKevin B Teuscher, Min Zhang, Haitao JiJournal of Medicinal Chemistry|July 16, 2021
Discovery of 1-Benzoyl 4-Phenoxypiperidines as Small-Molecule Inhibitors of the β-Catenin/B-Cell Lymphoma 9 Protein-Protein InteractionZilu Li, Min Zhang, Kevin B Teuscher, et al.ACS Medicinal Chemistry Letters|May 19, 2016
Structure-Based Design of 1,4-Dibenzoylpiperazines as β-Catenin/B-Cell Lymphoma 9 Protein-Protein Interaction InhibitorsJohn A Wisniewski, Jinya Yin, Kevin B Teuscher, et al.Journal of Medicinal Chemistry|October 1, 2021
Fragment-Based Discovery of Small Molecules Bound to T-Cell Immunoglobulin and Mucin Domain-Containing Molecule 3 (TIM-3)Tyson A Rietz, Kevin B Teuscher, Jonathan J Mills, et al.Journal of Medicinal Chemistry|April 18, 2022
Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based OptimizationKevin B Teuscher, Kenneth M Meyers, Qiangqiang Wei, et al.Journal of Medicinal Chemistry|February 2, 2026
Discovery of Spiro[chromane-2,4'-piperidine] Derivatives as Irreversible Inhibitors of SARS-CoV-2 Papain-like ProteaseQiangqiang Wei, Ashley J Taylor, Nagaraju Miriyala, et al.Journal of Medicinal Chemistry|December 12, 2023
Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 InhibitorsKevin B Teuscher, Jonathan J Mills, Jianhua Tian, et al.Proceedings of the National Academy of Sciences of the United States of America|August 21, 2024
Expanded profiling of WD repeat domain 5 inhibitors reveals actionable strategies for the treatment of hematologic malignanciesChristian T Meyer, Brianna N Smith, Jing Wang, et al.Pageof 2