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Bioorganic & Medicinal Chemistry Letters|December 11, 2012
Structure-activity relationship study on benzoic acid part of diphenylamine-based retinoidsKiminori Ohta, Emiko Kawachi, Koichi Shudo, et al.
International Journal of Molecular Sciences|February 15, 2022
Challenging Approach to the Development of Novel Estrogen Receptor Modulators Based on the Chemical Properties of GuaiazuleneKiminori Ohta, Asako Kaise, Takumi Ogawa, et al.
Bioorganic & Medicinal Chemistry Letters|November 26, 2013
Enhanced estrogen receptor beta (ERβ) selectivity of fluorinated carborane-containing ER modulatorsKiminori Ohta, Takumi Ogawa, Asako Kaise, et al.
Bioorganic & Medicinal Chemistry|May 20, 2014
Novel estrogen receptor (ER) modulators containing various hydrophobic bent-core structuresKiminori Ohta, Takumi Ogawa, Asako Kaise, et al.
Bioorganic & Medicinal Chemistry|December 25, 2017
Synthesis, structure-activity relationships, and mechanistic studies of 5-arylazo-tropolone derivatives as novel xanthine oxidase (XO) inhibitorsDaisuke Sato, Takuya Kisen, Mina Kumagai, et al.
Bioorganic & Medicinal Chemistry|January 24, 2015
Structure-activity relationship study of diphenylamine-based estrogen receptor (ER) antagonistsKiminori Ohta, Yuki Chiba, Asako Kaise, et al.
Bioorganic & Medicinal Chemistry Letters|June 17, 2015
Synthesis and biological evaluation of novel m-carborane-containing estrogen receptor partial agonists as SERM candidatesKiminori Ohta, Takumi Ogawa, Asako Kaise, et al.
Journal of Medicinal Chemistry|June 10, 2005
Potent estrogen receptor ligands based on bisphenols with a globular hydrophobic coreYasuyuki Endo, Tomohiro Yoshimi, Kiminori Ohta, et al.
Bioorganic & Medicinal Chemistry Letters|June 29, 2019
ER subtype selectivity of m-carborane-containing phenols: C-alkyl groups on the m-carborane cage enhance ERα selectivityKiminori Ohta, Takumi Ogawa, Koichi Kato, et al.
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