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Journal of Medicinal Chemistry|September 14, 2007
4-[omega-[4-arylpiperazin-1-yl]alkoxy]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualizationMarcello Leopoldo, Enza Lacivita, Elena Passafiume, et al.Chemmedchem|November 12, 2010
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Δ(8)-Δ(7) sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activityCarmen Abate, Mauro Niso, Marialessandra Contino, et al.Archiv Der Pharmazie|January 12, 2016
Functionalized Coumarine Fragment to Obtain Fluorescent and Selective P-Glycoprotein LigandsElena Capparelli, Marialessandra Contino, Maria G Perrone, et al.Pharmacology Research & Perspectives|October 31, 2015
Inhibition of hERG potassium channel by the antiarrhythmic agent mexiletine and its metabolite m-hydroxymexiletineRoberta Gualdani, Francesco Tadini-Buoninsegni, Mariagrazia Roselli, et al.Journal of Medicinal Chemistry|December 22, 2005
Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptorFrancesco Berardi, Savina Ferorelli, Carmen Abate, et al.Chemmedchem|January 23, 2016
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump OverexpressionStefano Guglielmo, Marialessandra Contino, Loretta Lazzarato, et al.European Journal of Medicinal Chemistry|December 3, 2014
From mixed sigma-2 receptor/P-glycoprotein targeting agents to selective P-glycoprotein modulators: small structural changes address the mechanism of interaction at the efflux pumpCarmen Abate, Maria Laura Pati, Marialessandra Contino, et al.Bioorganic & Medicinal Chemistry|November 15, 2011
Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities as σ₁ receptor ligandsSavina Ferorelli, Carmen Abate, Maria P Pedone, et al.Bioorganic & Medicinal Chemistry Letters|February 5, 2013
Potent and selective tariquidar bioisosters as potential PET radiotracers for imaging P-gpMarialessandra Contino, Laura Zinzi, Maria Grazia Perrone, et al.Journal of Medicinal Chemistry|December 14, 2004
Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agentsMarcello Leopoldo, Francesco Berardi, Nicola A Colabufo, et al.Pageof 12