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Bioorganic & Medicinal Chemistry Letters|February 15, 2002
Encounter with unexpected collagenase-1 selective inhibitor: switchover of inhibitor binding pocket induced by fluorine atomMasaaki Sawa, Hirosato Kondo, Shin-ichiro NishimuraBioorganic & Medicinal Chemistry Letters|December 5, 2017
Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitorsWataru Kawahata, Tokiko Asami, Takayuki Irie, et al.Journal of Medicinal Chemistry|February 8, 2002
A three-dimensional quantitative structure-activity relationship study of heparin-binding epidermal growth factor shedding inhibitors using comparative molecular field analysisRoberta Bursi, Masaaki Sawa, Yasuyuki Hiramatsu, et al.Bioorganic & Medicinal Chemistry Letters|April 7, 2015
'Turn On/Off' fluorescence probe for the screening of unactivated Bruton's tyrosine kinaseWataru Kawahata, Tokiko Asami, Ikuo Fujii, et al.Bioorganic & Medicinal Chemistry Letters|May 16, 2025
The discrepancies in amino acid sequence of the phosphate-binding loop lead to distinctive binding modes of a covalent inhibitor for MAP2K1 and MAP2K6: Structural insights for producing selective inhibitorsSeigo Yumura, Kei Moritsugu, Daisuke Kitagawa, et al.Bioorganic & Medicinal Chemistry Letters|June 5, 2003
Discovery of selective phosphonamide-based inhibitors of tumor necrosis factor-alpha converting enzyme (TACE)Masaaki Sawa, Kiriko Kurokawa, Yoshimasa Inoue, et al.Bioorganic & Medicinal Chemistry Letters|April 23, 2021
Identification of an allosteric and Smad3-selective inhibitor of p38αMAPK using a substrate-based approachHaruna Nagao, Daisuke Kitagawa, Fumio Nakajima, et al.Bioorganic & Medicinal Chemistry Letters|August 6, 2023
Low entropic cost of binding confers high selectivity on an allosteric ERK2 inhibitorHajime Sugiyama, Mayu Yoshida, Haruna Nagao, et al.Acta Crystallographica. Section F, Structural Biology Communications|July 9, 2019
A promiscuous kinase inhibitor delineates the conspicuous structural features of protein kinase CK2a1Masato Tsuyuguchi, Tetsuko Nakaniwa, Masaaki Sawa, et al.Biochemical and Biophysical Research Communications|January 22, 2022
Identification of a novel target site for ATP-independent ERK2 inhibitorsMayu Yoshida, Haruna Nagao, Hajime Sugiyama, et al.Pageof 7