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ACS Chemical Biology|November 19, 2015
SR2067 Reveals a Unique Kinetic and Structural Signature for PPARγ Partial AgonismLaura M van Marrewijk, Steven W Polyak, Marcel Hijnen, et al.Journal of Medicinal Chemistry|May 10, 2017
Structure-Activity Relationship of 2,4-Dichloro-N-(3,5-dichloro-4-(quinolin-3-yloxy)phenyl)benzenesulfonamide (INT131) Analogs for PPARγ-Targeted AntidiabeticsRebecca L Frkic, Yuanjun He, Beatriz B Rodriguez, et al.Elife|June 8, 2019
HDX-MS reveals structural determinants for RORγ hyperactivation by synthetic agonistsTimothy S Strutzenberg, Ruben D Garcia-Ordonez, Scott J Novick, et al.Bioorganic & Medicinal Chemistry Letters|August 26, 2018
Identification of potent RORβ modulators: Scaffold variationChristelle Doebelin, Rémi Patouret, Ruben D Garcia-Ordonez, et al.Journal of Molecular Biology|September 21, 2021
Conformational Changes of RORγ During Response Element Recognition and Coregulator EngagementTimothy S Strutzenberg, Yingmin Zhu, Scott J Novick, et al.Molecular Pharmacology|December 5, 2014
Antiproliferation activity of a small molecule repressor of liver receptor homolog 1Cesar A Corzo, Yelenis Mari, Mi Ra Chang, et al.ACS Chemical Biology|April 6, 2019
Unique Polypharmacology Nuclear Receptor Modulator Blocks Inflammatory Signaling PathwaysMi Ra Chang, Anthony Ciesla, Timothy S Strutzenberg, et al.Structure (London, England : 1993)|August 28, 2018
Chemical Crosslinking Mass Spectrometry Reveals the Conformational Landscape of the Activation Helix of PPARγ; a Model for Ligand-Dependent AntagonismJie Zheng, Cesar Corzo, Mi Ra Chang, et al.Chemmedchem|November 24, 2016
N-Arylsulfonyl Indolines as Retinoic Acid Receptor-Related Orphan Receptor γ (RORγ) AgonistsChristelle Doebelin, Rémi Patouret, Ruben D Garcia-Ordonez, et al.Structure (London, England : 1993)|January 17, 2012
Ligand and receptor dynamics contribute to the mechanism of graded PPARγ agonismTravis S Hughes, Michael J Chalmers, Scott Novick, et al.Pageof 24