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Bioorganic & Medicinal Chemistry|March 25, 2015
Structure-activity relationships of benzhydrol derivatives based on 1'-acetoxychavicol acetate (ACA) and their inhibitory activities on multiple myeloma cell growth via inactivation of the NF-κB pathwayTakashi Misawa, Kosuke Dodo, Minoru Ishikawa, et al.Chemical Communications (Cambridge, England)|August 6, 2025
Phthalimide: a potential warhead for switchable and bioorthogonal conjugationKosuke Chiba, Takumi Yoshida, Kana Okada, et al.Chemical Communications (Cambridge, England)|July 21, 2017
Specific fluorescence labeling of target proteins by using a ligand-4-azidophthalimide conjugateKosuke Chiba, Miwako Asanuma, Minoru Ishikawa, et al.Bioorganic & Medicinal Chemistry|November 29, 2005
Tricyclic pharmacophore-based molecules as novel integrin alpha(v)beta3 antagonists. Part 1: design and synthesis of a lead compound exhibiting alpha(v)beta3/alpha(IIb)beta3 dual antagonistic activityDai Kubota, Minoru Ishikawa, Mikio Yamamoto, et al.Bioorganic & Medicinal Chemistry Letters|June 18, 2013
Structure-activity relationships of bisphenol A analogs at estrogen receptors (ERs): discovery of an ERα-selective antagonistKeisuke Maruyama, Masaharu Nakamura, Shusuke Tomoshige, et al.Scientific Reports|June 17, 2021
Improvement in aqueous solubility of achiral symmetric cyclofenil by modification to a chiral asymmetric analogJunki Morimoto, Kazunori Miyamoto, Yuki Ichikawa, et al.Bioorganic & Medicinal Chemistry|April 8, 2014
Structure-activity relationship-guided development of retinoic acid receptor-related orphan receptor gamma (RORγ)-selective inverse agonists with a phenanthridin-6(5H)-one skeleton from a liver X receptor ligandYuko Nishiyama, Masahiko Nakamura, Takashi Misawa, et al.ACS Medicinal Chemistry Letters|July 24, 2018
Novel Nonsteroidal Progesterone Receptor (PR) Antagonists with a Phenanthridinone SkeletonYuko Nishiyama, Shuichi Mori, Makoto Makishima, et al.Bioorganic & Medicinal Chemistry|September 14, 2016
Structure-activity relationship studies of non-carboxylic acid peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonistsShogo Okazaki, Ryuta Shioi, Tomomi Noguchi-Yachide, et al.Bioorganic & Medicinal Chemistry Letters|May 26, 2017
Switching subtype-selectivity: Fragment replacement strategy affords novel class of peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonistsRyuta Shioi, Shogo Okazaki, Tomomi Noguchi-Yachide, et al.Pageof 8