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Nature Communications
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April 14, 2025
Drugit: crowd-sourcing molecular design of non-peptidic VHL binders
Thomas Scott, Christian Alan Paul Smethurst, Yvonne Westermaier, et al.
Journal of Medicinal Chemistry
|
October 27, 2022
Fragment Optimization of Reversible Binding to the Switch II Pocket on KRAS Leads to a Potent, In Vivo Active KRAS<sup>G12C</sup> Inhibitor
Joachim Bröker, Alex G Waterson, Chris Smethurst, et al.
Journal of Medicinal Chemistry
|
July 25, 2025
Discovery of BI-2493, a Pan-KRAS Inhibitor Showing <i>In Vivo</i> Efficacy
Joachim Bröker, Alex G Waterson, Timothy R Hodges, et al.
Chemmedchem
|
December 4, 2020
Getting a Grip on the Undrugged: Targeting β-Catenin with Fragment-Based Methods
Dirk Kessler, Moriz Mayer, Stephan K Zahn, et al.
Nature Communications
|
October 10, 2022
A selective and orally bioavailable VHL-recruiting PROTAC achieves SMARCA2 degradation in vivo
Christiane Kofink, Nicole Trainor, Barbara Mair, et al.
Journal of Medicinal Chemistry
|
November 6, 2019
Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors
Harald Engelhardt, Dietrich Böse, Mark Petronczki, et al.
Journal of Medicinal Chemistry
|
August 1, 2019
Intracellular Trapping of the Selective Phosphoglycerate Dehydrogenase (PHGDH) Inhibitor <b>BI-4924</b> Disrupts Serine Biosynthesis
Harald Weinstabl, Matthias Treu, Joerg Rinnenthal, et al.
Proceedings of the National Academy of Sciences of the United States of America
|
February 13, 2020
Reply to Tran et al.: Dimeric KRAS protein-protein interaction stabilizers
Dirk Kessler, Andreas Gollner, Michael Gmachl, et al.
Proceedings of the National Academy of Sciences of the United States of America
|
July 24, 2019
Drugging an undruggable pocket on KRAS
Dirk Kessler, Michael Gmachl, Andreas Mantoulidis, et al.
Cell Reports
|
September 21, 2017
Chemically Induced Degradation of the Oncogenic Transcription Factor BCL6
Nina Kerres, Steffen Steurer, Stefanie Schlager, et al.
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Search research articles
Search
Showing results (21-30 of 31) with videos related to
Sort By:
Page
of 4
Nature Communications
|
April 14, 2025
Drugit: crowd-sourcing molecular design of non-peptidic VHL binders
Thomas Scott, Christian Alan Paul Smethurst, Yvonne Westermaier, et al.
Journal of Medicinal Chemistry
|
October 27, 2022
Fragment Optimization of Reversible Binding to the Switch II Pocket on KRAS Leads to a Potent, In Vivo Active KRAS<sup>G12C</sup> Inhibitor
Joachim Bröker, Alex G Waterson, Chris Smethurst, et al.
Journal of Medicinal Chemistry
|
July 25, 2025
Discovery of BI-2493, a Pan-KRAS Inhibitor Showing <i>In Vivo</i> Efficacy
Joachim Bröker, Alex G Waterson, Timothy R Hodges, et al.
Chemmedchem
|
December 4, 2020
Getting a Grip on the Undrugged: Targeting β-Catenin with Fragment-Based Methods
Dirk Kessler, Moriz Mayer, Stephan K Zahn, et al.
Nature Communications
|
October 10, 2022
A selective and orally bioavailable VHL-recruiting PROTAC achieves SMARCA2 degradation in vivo
Christiane Kofink, Nicole Trainor, Barbara Mair, et al.
Journal of Medicinal Chemistry
|
November 6, 2019
Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors
Harald Engelhardt, Dietrich Böse, Mark Petronczki, et al.
Journal of Medicinal Chemistry
|
August 1, 2019
Intracellular Trapping of the Selective Phosphoglycerate Dehydrogenase (PHGDH) Inhibitor <b>BI-4924</b> Disrupts Serine Biosynthesis
Harald Weinstabl, Matthias Treu, Joerg Rinnenthal, et al.
Proceedings of the National Academy of Sciences of the United States of America
|
February 13, 2020
Reply to Tran et al.: Dimeric KRAS protein-protein interaction stabilizers
Dirk Kessler, Andreas Gollner, Michael Gmachl, et al.
Proceedings of the National Academy of Sciences of the United States of America
|
July 24, 2019
Drugging an undruggable pocket on KRAS
Dirk Kessler, Michael Gmachl, Andreas Mantoulidis, et al.
Cell Reports
|
September 21, 2017
Chemically Induced Degradation of the Oncogenic Transcription Factor BCL6
Nina Kerres, Steffen Steurer, Stefanie Schlager, et al.
Page
of 4