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P Caldwell

Showing results (121-130 of 132) with videos related to

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Bioorganic & Medicinal Chemistry Letters|December 3, 2014
Discovery of potent iminoheterocycle BACE1 inhibitorsJohn P Caldwell, Robert D Mazzola, James Durkin, et al.
Chembiochem : a European Journal of Chemical Biology|February 1, 2020
Cyp1 Inhibition Prevents Doxorubicin-Induced Cardiomyopathy in a Zebrafish Heart-Failure ModelPui-Ying Lam, Peter Kutchukian, Rajan Anand, et al.
Bioorganic & Medicinal Chemistry Letters|August 21, 2010
Iminoheterocycles as gamma-secretase modulatorsJohn P Caldwell, Chad E Bennett, Troy M McCracken, et al.
Bioorganic & Medicinal Chemistry Letters|April 3, 2009
The discovery of tropane derivatives as nociceptin receptor ligands for the management of cough and anxietyGinny D Ho, John Anthes, Ana Bercovici, et al.
Journal of Medicinal Chemistry|November 3, 2018
Overcoming Time-Dependent Inhibition (TDI) of Cytochrome P450 3A4 (CYP3A4) Resulting from Bioactivation of a Fluoropyrimidine MoietyMihirbaran Mandal, Kaushik Mitra, Diane Grotz, et al.
Journal of Medicinal Chemistry|September 20, 2012
Design and validation of bicyclic iminopyrimidinones as beta amyloid cleaving enzyme-1 (BACE1) inhibitors: conformational constraint to favor a bioactive conformationMihirbaran Mandal, Zhaoning Zhu, Jared N Cumming, et al.
Bioorganic & Medicinal Chemistry Letters|March 3, 2015
Iminopyrimidinones: a novel pharmacophore for the development of orally active renin inhibitorsBrian A McKittrick, John P Caldwell, Thomas Bara, et al.
Journal of Medicinal Chemistry|March 4, 2016
Structure-Based Design of an Iminoheterocyclic β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE) Inhibitor that Lowers Central Aβ in Nonhuman PrimatesMihirbaran Mandal, Yusheng Wu, Jeffrey Misiaszek, et al.
ACS Medicinal Chemistry Letters|April 15, 2026
DNA-Encoded Library (DEL) Selection Identifies a Distinct DDB1 Ligand Binding SiteShiva Krishna Reddy Guduru, John P Caldwell, Katherine M Digianantonio, et al.
Journal of Medicinal Chemistry|March 22, 2017
Can We Make Small Molecules Lean? Optimization of a Highly Lipophilic TarO InhibitorMihirbaran Mandal, Zheng Tan, Christina Madsen-Duggan, et al.
Pageof 14

Showing results (121-130 of 132) with videos related to

Sort By:
Pageof 14
Bioorganic & Medicinal Chemistry Letters|December 3, 2014
Discovery of potent iminoheterocycle BACE1 inhibitorsJohn P Caldwell, Robert D Mazzola, James Durkin, et al.
Chembiochem : a European Journal of Chemical Biology|February 1, 2020
Cyp1 Inhibition Prevents Doxorubicin-Induced Cardiomyopathy in a Zebrafish Heart-Failure ModelPui-Ying Lam, Peter Kutchukian, Rajan Anand, et al.
Bioorganic & Medicinal Chemistry Letters|August 21, 2010
Iminoheterocycles as gamma-secretase modulatorsJohn P Caldwell, Chad E Bennett, Troy M McCracken, et al.
Bioorganic & Medicinal Chemistry Letters|April 3, 2009
The discovery of tropane derivatives as nociceptin receptor ligands for the management of cough and anxietyGinny D Ho, John Anthes, Ana Bercovici, et al.
Journal of Medicinal Chemistry|November 3, 2018
Overcoming Time-Dependent Inhibition (TDI) of Cytochrome P450 3A4 (CYP3A4) Resulting from Bioactivation of a Fluoropyrimidine MoietyMihirbaran Mandal, Kaushik Mitra, Diane Grotz, et al.
Journal of Medicinal Chemistry|September 20, 2012
Design and validation of bicyclic iminopyrimidinones as beta amyloid cleaving enzyme-1 (BACE1) inhibitors: conformational constraint to favor a bioactive conformationMihirbaran Mandal, Zhaoning Zhu, Jared N Cumming, et al.
Bioorganic & Medicinal Chemistry Letters|March 3, 2015
Iminopyrimidinones: a novel pharmacophore for the development of orally active renin inhibitorsBrian A McKittrick, John P Caldwell, Thomas Bara, et al.
Journal of Medicinal Chemistry|March 4, 2016
Structure-Based Design of an Iminoheterocyclic β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE) Inhibitor that Lowers Central Aβ in Nonhuman PrimatesMihirbaran Mandal, Yusheng Wu, Jeffrey Misiaszek, et al.
ACS Medicinal Chemistry Letters|April 15, 2026
DNA-Encoded Library (DEL) Selection Identifies a Distinct DDB1 Ligand Binding SiteShiva Krishna Reddy Guduru, John P Caldwell, Katherine M Digianantonio, et al.
Journal of Medicinal Chemistry|March 22, 2017
Can We Make Small Molecules Lean? Optimization of a Highly Lipophilic TarO InhibitorMihirbaran Mandal, Zheng Tan, Christina Madsen-Duggan, et al.
Pageof 14