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Paul Brear

Showing results (31-40 of 41) with videos related to

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Journal of Medicinal Chemistry|July 11, 2023
Structure-Guided Chemical Optimization of Bicyclic Peptide (<i>Bicycle</i>) Inhibitors of Angiotensin-Converting Enzyme 2Maximilian A J Harman, Steven J Stanway, Heather Scott, et al.
European Journal of Medicinal Chemistry|March 15, 2022
Anthraquinone derivatives as ADP-competitive inhibitors of liver pyruvate kinaseAmalyn Nain-Perez, Anders Foller Füchtbauer, Liliana Håversen, et al.
Nature Chemical Biology|October 31, 2023
Chemical proteomics reveals the target landscape of 1,000 kinase inhibitorsMaria Reinecke, Paul Brear, Larsen Vornholz, et al.
Scientific Reports|November 6, 2019
Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitorsIrina Kufareva, Benoit Bestgen, Paul Brear, et al.
Journal of Medicinal Chemistry|March 24, 2026
Yeast Display Technology Enables Rapid Discovery of Low-Nanomolar Macrocyclic Peptide Inhibitors of Human Angiotensin-Converting Enzyme 2Zhanna Romanyuk, Giacomo Bettin, Paul Brear, et al.
Iscience|May 6, 2026
Two birds with one stone: An antibiotic hit blocking <i>Staphylococcus aureus</i> heme uptake with serendipitous hemoglobin left-shifting activitySarah Hijazi, Francesco Marchesani, Marialaura Marchetti, et al.
ACS Nano|February 13, 2026
Utilizing Constrained Bicyclic Peptides for <i>In Vitro</i> DiagnosticsAndré Shamsabadi, Adam Creamer, Christy J Sadler, et al.
Chemistry & Biology|July 31, 2012
ALDH2 mediates 5-nitrofuran activity in multiple speciesLinna Zhou, Hironori Ishizaki, Michaela Spitzer, et al.
Nature Biotechnology|August 14, 2024
Rapid discovery of monoclonal antibodies by microfluidics-enabled FACS of single pathogen-specific antibody-secreting cellsKatrin Fischer, Aleksei Lulla, Tsz Y So, et al.
Chemical Science|June 7, 2021
Demonstration of the utility of DOS-derived fragment libraries for rapid hit derivatisation in a multidirectional fashionSarah L Kidd, Elaine Fowler, Till Reinhardt, et al.
Pageof 5

Showing results (31-40 of 41) with videos related to

Sort By:
Pageof 5
Journal of Medicinal Chemistry|July 11, 2023
Structure-Guided Chemical Optimization of Bicyclic Peptide (<i>Bicycle</i>) Inhibitors of Angiotensin-Converting Enzyme 2Maximilian A J Harman, Steven J Stanway, Heather Scott, et al.
European Journal of Medicinal Chemistry|March 15, 2022
Anthraquinone derivatives as ADP-competitive inhibitors of liver pyruvate kinaseAmalyn Nain-Perez, Anders Foller Füchtbauer, Liliana Håversen, et al.
Nature Chemical Biology|October 31, 2023
Chemical proteomics reveals the target landscape of 1,000 kinase inhibitorsMaria Reinecke, Paul Brear, Larsen Vornholz, et al.
Scientific Reports|November 6, 2019
Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitorsIrina Kufareva, Benoit Bestgen, Paul Brear, et al.
Journal of Medicinal Chemistry|March 24, 2026
Yeast Display Technology Enables Rapid Discovery of Low-Nanomolar Macrocyclic Peptide Inhibitors of Human Angiotensin-Converting Enzyme 2Zhanna Romanyuk, Giacomo Bettin, Paul Brear, et al.
Iscience|May 6, 2026
Two birds with one stone: An antibiotic hit blocking <i>Staphylococcus aureus</i> heme uptake with serendipitous hemoglobin left-shifting activitySarah Hijazi, Francesco Marchesani, Marialaura Marchetti, et al.
ACS Nano|February 13, 2026
Utilizing Constrained Bicyclic Peptides for <i>In Vitro</i> DiagnosticsAndré Shamsabadi, Adam Creamer, Christy J Sadler, et al.
Chemistry & Biology|July 31, 2012
ALDH2 mediates 5-nitrofuran activity in multiple speciesLinna Zhou, Hironori Ishizaki, Michaela Spitzer, et al.
Nature Biotechnology|August 14, 2024
Rapid discovery of monoclonal antibodies by microfluidics-enabled FACS of single pathogen-specific antibody-secreting cellsKatrin Fischer, Aleksei Lulla, Tsz Y So, et al.
Chemical Science|June 7, 2021
Demonstration of the utility of DOS-derived fragment libraries for rapid hit derivatisation in a multidirectional fashionSarah L Kidd, Elaine Fowler, Till Reinhardt, et al.
Pageof 5