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Bioorganic & Medicinal Chemistry Letters|February 9, 2010
Discovery of N-(5,6-diarylpyridin-2-yl)amide derivatives as potent and selective A(2B) adenosine receptor antagonistsPaul Eastwood, Jacob Gonzalez, Sergio Paredes, et al.Bioorganic & Medicinal Chemistry Letters|August 5, 2011
Indolin-2-one p38α inhibitors II: Lead optimisationPaul Eastwood, Jacob González, Elena Gómez, et al.Bioorganic & Medicinal Chemistry Letters|June 24, 2011
Indolin-2-one p38α inhibitors I: design, profiling and crystallographic binding modePaul Eastwood, Jacob González, Elena Gómez, et al.Bioorganic & Medicinal Chemistry Letters|October 1, 2011
Indolin-2-one p38α inhibitors III: bioisosteric amide replacementPaul Eastwood, Jacob González, Elena Gómez, et al.Bioorganic & Medicinal Chemistry Letters|February 9, 2010
Discovery of potent and selective bicyclic A(2B) adenosine receptor antagonists via bioisosteric amide replacementPaul Eastwood, Jacob Gonzalez, Sergio Paredes, et al.Bioorganic & Medicinal Chemistry Letters|April 24, 2012
Novel triazolopyridylbenzamides as potent and selective p38α inhibitorsJosep Aiguadé, Cristina Balagué, Inés Carranco, et al.Plos One|January 11, 2018
Application of a phenotypic drug discovery strategy to identify biological and chemical starting points for inhibition of TSLP production in lung epithelial cellsAdelina Orellana, Vicente García-González, Rosa López, et al.ACS Medicinal Chemistry Letters|June 6, 2014
Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor AntagonistPaul Eastwood, Cristina Esteve, Jacob González, et al.Journal of Medicinal Chemistry|October 15, 2019
Identification of 2-Imidazopyridine and 2-Aminopyridone Purinones as Potent Pan-Janus Kinase (JAK) Inhibitors for the Inhaled Treatment of Respiratory DiseasesJordi Bach, Paul Eastwood, Jacob González, et al.Bioorganic & Medicinal Chemistry Letters|August 28, 2003
Mapping the kinase domain of Janus Kinase 3Christopher Adams, David J Aldous, Shelley Amendola, et al.Pageof 2