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Drug Development Research|May 27, 2026
Lead Discovery via Scaffold Refinement: Structure-Guided Optimization of 1,2,4-Triazolo[1,5-a]Pyrimidines as Potent Dual EGFR/CDK-2 Inhibitors Targeting Colorectal CarcinomaRowida Nasr, Hesham Haffez, Mohamed S Nafie, et al.Archiv Der Pharmazie|July 17, 2026
Thiazole-Derived Dual EGFR/CDK-2 Inhibitors: Rational Design, Synthesis, In Vitro Anticancer Evaluation, Mechanistic Profiling, and Computational Binding AnalysisRowida Nasr, Mohamed S Nafie, Hesham Haffez, et al.Pageof 1