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Psychoneuroendocrinology|August 24, 2010
Anxiolytic properties of a 2-phenylindolglyoxylamide TSPO ligand: Stimulation of in vitro neurosteroid production affecting GABAA receptor activityBarbara Costa, Eleonora Da Pozzo, Beatrice Chelli, et al.Journal of Medicinal Chemistry|March 19, 2004
N,N-dialkyl-2-phenylindol-3-ylglyoxylamides. A new class of potent and selective ligands at the peripheral benzodiazepine receptorGiampaolo Primofiore, Federico Da Settimo, Sabrina Taliani, et al.Molecular Neurobiology|January 12, 2022
Translocator Protein Ligand PIGA1138 Reduces Disease Symptoms and Severity in Experimental Autoimmune Encephalomyelitis Model of Primary Progressive Multiple SclerosisChiara Tremolanti, Chiara Cavallini, Laurence Meyer, et al.Dalton Transactions (Cambridge, England : 2003)|June 23, 2021
Two mixed valence diruthenium(II,III) isomeric complexes show different anticancer propertiesElisabetta Barresi, Iogann Tolbatov, Tiziano Marzo, et al.Biochimica Et Biophysica Acta. Molecular Basis of Disease|April 30, 2026
18 kDa TSPO-mediated neurosteroidogenesis controls cholesterol homeostasis in tuning microglia response to inflammatory stimulusElisa Angeloni, Lorenzo Germelli, Laura Marchetti, et al.European Journal of Medicinal Chemistry|April 30, 2026
Recent advances in the development of selective hMAO-B inhibitors for neurodegenerative diseases: An update from 2020 to presentSilvia Salerno, Giovanni Fabbri, Maria Luisa Di Paolo, et al.Journal of Chemical Information and Modeling|September 14, 2024
Discovering Dually Active Anti-cancer Compounds with a Hybrid AI-structure-based ApproachMichele Roggia, Benito Natale, Giorgio Amendola, et al.Archiv Der Pharmazie|July 29, 2022
New antiproliferative agents derived from tricyclic 3,4-dihydrobenzo[4,5]imidazo[1,2-a][1,3,5]triazine scaffold: Synthesis and pharmacological effectsMarco Robello, Silvia Salerno, Elisabetta Barresi, et al.Journal of Medicinal Chemistry|August 5, 2005
Novel, highly potent adenosine deaminase inhibitors containing the pyrazolo[3,4-d]pyrimidine ring system. Synthesis, structure-activity relationships, and molecular modeling studiesFederico Da Settimo, Giampaolo Primofiore, Concettina La Motta, et al.Journal of Medicinal Chemistry|June 19, 2018
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX InhibitorsSilvia Salerno, Elisabetta Barresi, Giorgio Amendola, et al.Pageof 14