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Biochemical Pharmacology|May 21, 2011
Effects of highly active novel artemisinin-chloroquinoline hybrid compounds on β-hematin formation, parasite morphology and endocytosis in Plasmodium falciparumTzu-Shean Feng, Eric M Guantai, Margo Nell, et al.Bioorganic & Medicinal Chemistry Letters|March 8, 2011
Novel thiolactone-isatin hybrids as potential antimalarial and antitubercular agentsRenate H Hans, Ian J F Wiid, Paul D van Helden, et al.Bioorganic & Medicinal Chemistry|July 31, 2013
Tetrazole-based deoxyamodiaquines: synthesis, ADME/PK profiling and pharmacological evaluation as potential antimalarial agentsMatshawandile Tukulula, Mathew Njoroge, Grace C Mugumbate, et al.Journal of Medicinal Chemistry|February 3, 2022
Probing the Requirements for Dual Angiotensin-Converting Enzyme C-Domain Selective/Neprilysin InhibitionLauren B Arendse, Gyles E Cozier, Charles J Eyermann, et al.ACS Medicinal Chemistry Letters|August 20, 2021
Structure-Activity Relationship Studies Reveal New Astemizole Analogues Active against Plasmodium falciparum In VitroDickson Mambwe, Malkeet Kumar, Richard Ferger, et al.Journal of Medicinal Chemistry|April 1, 2025
Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin InhibitorsGyles E Cozier, Lauren B Coulson, Charles J Eyermann, et al.ACS Infectious Diseases|July 17, 2019
Semisynthetic Antimycobacterial C-3 Silicate and C-3/C-21 Ester Derivatives of Fusidic Acid: Pharmacological Evaluation and Stability Studies in Liver Microsomes, Rat Plasma, and Mycobacterium tuberculosis cultureMathew Njoroge, Gurminder Kaur, Marlene Espinoza-Moraga, et al.Bioorganic & Medicinal Chemistry Letters|January 5, 2010
Synthesis, antimalarial and antitubercular activity of acetylenic chalconesRenate H Hans, Eric M Guantai, Carmen Lategan, et al.Journal of Medicinal Chemistry|May 28, 2004
Synthesis and structure-activity relationships of parasiticidal thiosemicarbazone cysteine protease inhibitors against Plasmodium falciparum, Trypanosoma brucei, and Trypanosoma cruziDoron C Greenbaum, Zachary Mackey, Elizabeth Hansell, et al.Bioorganic & Medicinal Chemistry|August 13, 2015
Antimalarial benzoheterocyclic 4-aminoquinolines: Structure-activity relationship, in vivo evaluation, mechanistic and bioactivation studiesDennis S B Ongarora, Natasha Strydom, Kathryn Wicht, et al.Pageof 31