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ACS Medicinal Chemistry Letters|July 16, 2021
Discovery of Potent Selective Nonzinc Binding Autotaxin Inhibitor BIO-32546Bin Ma, Lei Zhang, Lihong Sun, et al.
ACS Medicinal Chemistry Letters|July 16, 2021
Discovery and Optimization of a Series of Benzofuran Selective ERAP1 Inhibitors: Biochemical and In Silico StudiesSafia Deddouche-Grass, Cyrielle Andouche, Felix Bärenz, et al.
ACS Medicinal Chemistry Letters|July 16, 2021
Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 InhibitorsEmily C Cherney, Liping Zhang, Weiwei Guo, et al.
ACS Medicinal Chemistry Letters|July 16, 2021
DNA-Encoded Library Hit Confirmation: Bridging the Gap Between On-DNA and Off-DNA ChemistryBing Xia, G Joseph Franklin, Xiaojie Lu, et al.
ACS Medicinal Chemistry Letters|July 16, 2021
Design and Synthesis of TRAP1 Selective Inhibitors: H-Bonding with Asn171 Residue in TRAP1 Increases Paralog SelectivitySujae Yang, Nam Gu Yoon, Dongyoung Kim, et al.
ACS Medicinal Chemistry Letters|June 17, 2021
Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as StabilizersEline Sijbesma, Kenneth K Hallenbeck, Sebastian A Andrei, et al.
ACS Medicinal Chemistry Letters|June 18, 2021
Remodelin Is a Cryptic Assay Interference Chemotype That Does Not Inhibit NAT10-Dependent Cytidine AcetylationJonathan H Shrimp, Yihang Jing, Supuni Thalalla Gamage, et al.
ACS Medicinal Chemistry Letters|June 18, 2021
Mining for Ligandable Cavities in RNAJingru Xie, Aaron T Frank
ACS Medicinal Chemistry Letters|June 18, 2021
Discovery of Potent, Selective Triazolothiadiazole-Containing c-Met InhibitorsQing Tang, Alex M Aronov, David D Deininger, et al.
ACS Medicinal Chemistry Letters|June 18, 2021
Discovery of Orally Bioavailable Ligand Efficient Quinazolindiones as Potent and Selective Tankyrases InhibitorsDonghui Qin, Xiaojuan Lin, Zhi Liu, et al.
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