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ACS Medicinal Chemistry Letters|May 20, 2026
Computer-Aided Design of Plasmodium chabaudi-Derived Peptides with Dual Antibiofilm and Anti-inflammatory ActivitiesRaquel M Quigua Orozco, Alexandre D O Santos, Joelma P Rossetto, et al.ACS Medicinal Chemistry Letters|May 20, 2026
Lead Optimization of Xanthone Derivatives as Hepatitis B Virus cccDNA Reducers: Design, Synthesis, and BioevaluationLijun Guo, Xiaodong Chen, Xuejun Liu, et al.ACS Medicinal Chemistry Letters|May 20, 2026
DEL2PH4: Predictive 3D Pharmacophores from DNA-Encoded Library Screening DataMiklos Feher, Rebecca J Swett, Ryan T Walsh, et al.ACS Medicinal Chemistry Letters|May 20, 2026
Structural and Pharmacological Characterization of AT-121 Reveals Carbonic Anhydrase Inhibition as a Complementary Mechanism to Dual MOR/NOR AgonismAlessandro Bonardi, Marta Ferraroni, Paola Gratteri, et al.ACS Medicinal Chemistry Letters|May 20, 2026
Targeted Modulation of YAP Signaling: Advancing Small-Molecule Strategies in Oncology and Tissue RegenerationAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|May 20, 2026
Negatively Charged Pronucleotides as Inhibitors of Glioma Cell ProliferationJoanna Romanowska, Dariusz Wawrzyniak, Agnieszka Szymanska-Michalak, et al.ACS Medicinal Chemistry Letters|May 20, 2026
Novel Macrocyclic Compounds Targeting STING for Autoimmune Diseases TreatmentYanwei Jiang, Steven H LiangACS Medicinal Chemistry Letters|May 20, 2026
Spirocyclohexane-Chroman-4-one Derivatives as Selectively Cytotoxic Agents in Breast Cancer ModelsDaria A Ipatova, Viktoria A Ikonnikova, Kirill D Kungurtsev, et al.ACS Medicinal Chemistry Letters|May 20, 2026
Discovery and Optimization of Potent and Subtype-Selective Urea-Derived NaV1.8 InhibitorsClemens Dialer, Sebastian Krüger, Markus Wagener, et al.ACS Medicinal Chemistry Letters|May 26, 2018
Cyclic Peptidic Mimetics of Apollo Peptides Targeting Telomeric Repeat Binding Factor 2 (TRF2) and Apollo InteractionXia Chen, Liu Liu, Yong Chen, et al.Pageof 441