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ACS Medicinal Chemistry Letters|June 17, 2026
Synthesis and Biochemical Characterization of Investigational Pyrazolopyrimidine-Based Allosteric KRAS ModulatorsCynthia V Pagba, Kasuni Dilsha, Rakshya Ojha, et al.ACS Medicinal Chemistry Letters|June 17, 2026
Structure-Guided Discovery of Novel Highly Potent and Selective MTA-Cooperative PRMT5 InhibitorsChuping Huang, Min Liang, Ping Zhang, et al.ACS Medicinal Chemistry Letters|June 17, 2026
Structure-Based Search for Novel Creatine Transporter InhibitorsDorota Stary, Ali El-Kasaby, Danila Boytsov, et al.ACS Medicinal Chemistry Letters|June 17, 2026
Degrading Immune Checkpoints and Coordinating Oncogenic Signaling: Emerging Strategies in Cancer TherapyAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|June 17, 2026
Targeted Protein Degradation and Metabolic Inhibition as Complementary Therapeutic Strategies: TEAD PROTACs and NAT8L Inhibitors in OncologyAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|June 17, 2026
Solubility-Driven Lead Optimization of PAR4 Antagonists and Evaluation of a Phosphate Ester Prodrug Delivery StrategyO Scott Halpern, Samuel K Reznik, Xiaojun Zhang, et al.ACS Medicinal Chemistry Letters|June 17, 2026
Degradation and Detection: Integrating BCL6 Targeted Protein Degradation with Biomarker-Guided BET Inhibition in CancerAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|June 17, 2026
5‑Nitrofuran-Semicarbazone Hybrids as Antitrypanosomal Agents: Structure-Activity Relationship and Nitroreductase ActivationTemitayo O Alegbejo Price, Daniel G Silva, Miguel M Vaidergorn, et al.ACS Medicinal Chemistry Letters|June 17, 2026
4‑Aminoalkylquinolines as Potent Antitubercular Agents Targeting the Cytochrome bc1 ComplexEstevão Silveira Grams, Alessandro Silva Ramos, Fernanda Fries da Silva, et al.ACS Medicinal Chemistry Letters|June 17, 2026
Novel Tricyclic Compounds as 5‑HT2A Receptor Agonists for Treating Depression, Anxiety, Substance Abuse, and HeadachesRam W Sabnis, Anika R SabnisPageof 441