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Bioorganic & Medicinal Chemistry Letters|June 1, 2019
Discovery of conolidine derivative DS39201083 as a potent novel analgesic without mu opioid agonist activityTsuyoshi Arita, Masayoshi Asano, Kazufumi Kubota, et al.
Bioorganic & Medicinal Chemistry Letters|June 3, 2019
Discovery of naphthacemycins as a novel class of PARP1 inhibitorsWenbin Shen, Xinhua Lu, Jingtong Zhu, et al.
Bioorganic & Medicinal Chemistry Letters|June 5, 2019
Discovery of piperazic acid peptide deformylase inhibitors with in vivo activity for respiratory tract and skin infectionsJared T Spletstoser, Jason Dreabit, Andrew N Knox, et al.
Bioorganic & Medicinal Chemistry Letters|May 29, 2019
Influence of lysine residue in amphipathic helical peptides on targeted delivery of RNA into cancer cellsShun-Ichi Wada, Kohei Taniguchi, Hiroaki Hamazaki, et al.
Bioorganic & Medicinal Chemistry Letters|May 29, 2019
Discovery of ABT-957: 1-Benzyl-5-oxopyrrolidine-2-carboxamides as selective calpain inhibitors with enhanced metabolic stabilityKatja Jantos, Andreas Kling, Helmut Mack, et al.
Bioorganic & Medicinal Chemistry Letters|September 29, 2018
Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatmentAlessio Molinari, Anna Lucia Fallacara, Salvatore Di Maria, et al.
Bioorganic & Medicinal Chemistry Letters|September 30, 2018
Design, synthesis, and evaluation of carboxyl-modified oseltamivir derivatives with improved lipophilicity as neuraminidase inhibitorsBoyu Wang, Kuanglei Wang, Peipei Meng, et al.
Bioorganic & Medicinal Chemistry Letters|May 20, 2019
Design, synthesis and biological evaluation of benzimidazole derivatives as novel human Pin1 inhibitorsTianyi Ma, Min Huang, Aihua Li, et al.
Bioorganic & Medicinal Chemistry Letters|May 21, 2019
Synthesis and antiviral activity of coumarin derivatives against infectious hematopoietic necrosis virusYang Hu, Weichao Chen, Yufeng Shen, et al.
Bioorganic & Medicinal Chemistry Letters|May 4, 2019
Resistance mechanisms and cross-resistance for a pyridine-pyrimidine amide inhibitor of microtubule polymerizationJ Chancellor Fox, Alex T Evans, Michael P Blomfield, et al.
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