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Bioorganic & Medicinal Chemistry Letters|March 18, 2003
Synthesis of fluorescence-labeled sphingosine and sphingosine 1-phosphate; effective tools for sphingosine and sphingosine 1-phosphate behaviorToshikazu Hakogi, Toshihiko Shigenari, Shigeo Katsumura, et al.Bioorganic & Medicinal Chemistry Letters|March 18, 2003
Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-positive antibacterial activityRichard L Jarvest, John M Berge, Murray J Brown, et al.Bioorganic & Medicinal Chemistry Letters|March 18, 2003
Novel N1-(benzyl)cinnamamidine derived NR2B subtype-selective NMDA receptor antagonistsNeil R Curtis, Helen J Diggle, Janusz J Kulagowski, et al.Bioorganic & Medicinal Chemistry Letters|March 18, 2003
A structure-permeability study of small drug-like moleculesThomas Fichert, Mehran Yazdanian, John R ProudfootBioorganic & Medicinal Chemistry Letters|March 18, 2003
Binding of nicotine and homoazanicotine analogues at neuronal nicotinic acetylcholinergic (nACh) receptorsG Ferretti, M Dukat, M Giannella, et al.Bioorganic & Medicinal Chemistry Letters|March 18, 2003
Functional expression and characterization of EryA, the erythritol kinase of Brucella abortus, and enzymatic synthesis of L-erythritol-4-phosphateAntonietta M Lillo, Charles N Tetzlaff, Félix J Sangari, et al.Bioorganic & Medicinal Chemistry Letters|March 27, 2003
The inhibitory effects of squalene-derived triterpenes on protein phosphatase PP2AMaría L Souto, Claudia P Manríquez, Manuel Norte, et al.Bioorganic & Medicinal Chemistry Letters|March 27, 2003
Potent and selective aggrecanase inhibitors containing cyclic P1 substituentsRobert J Cherney, Ruowei Mo, Dayton T Meyer, et al.Bioorganic & Medicinal Chemistry Letters|March 27, 2003
Novel and potent human and rat beta3-adrenergic receptor agonists containing substituted 3-indolylalkylaminesHiroshi Harada, Yoshimi Hirokawa, Kenji Suzuki, et al.Bioorganic & Medicinal Chemistry Letters|March 27, 2003
Structure-activity relationship of cyclic peptide penta-c[Asp-His(6)-DPhe(7)-Arg(8)-Trp(9)-Lys]-NH(2) at the human melanocortin-1 and -4 receptors: His(6) substitutionAdrian Wai-Hing Cheung, Waleed Danho, Joseph Swistok, et al.Pageof 2,631