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European Journal of Medicinal Chemistry|January 24, 2025
Recent advances in small molecule design strategies against hepatic fibrosisHeming Chen, Wei Su, Tingting Li, et al.European Journal of Medicinal Chemistry|January 23, 2025
The development of α, β-unsaturated lactam-based andrographolide derivatives as anti-gastric cancer agents with the ability of inhibiting the ERK/c-Fos/Jun pathwayHang Zhang, Zhihao Xu, Zhengyu Xu, et al.European Journal of Medicinal Chemistry|January 17, 2025
A comparative study on the antioxidant and antiglycation properties of different vitamin D formsCezary Pawlukianiec, Kamil Klaudiusz Lauko, Daniel Michalak, et al.European Journal of Medicinal Chemistry|January 18, 2025
Discovery of novel capsaicin analogs as TRPV1 inhibitors for the treatment of idiopathic pulmonary fibrosisYu Cao, Yongju Wen, Zongyuan Zhou, et al.European Journal of Medicinal Chemistry|January 7, 2025
Discovery of 4,5-dihydro-benzo[g]indazole-based hydroxamic acids as HDAC3/BRD4 dual inhibitors and anti-tumor agentsBo Li, Yibing Chen, Siyuan Wang, et al.European Journal of Medicinal Chemistry|January 5, 2025
Correction of aberrant splicing of ELP1 pre-mRNA by kinetin derivatives - A structure activity relationship studyBarbara Maková, Václav Mik, Barbora Lišková, et al.European Journal of Medicinal Chemistry|December 29, 2024
Design, synthesis and biological evaluation of galantamine analogues for cognitive improvement in Alzheimer's diseaseMengzhen Li, Chao Ma, Yao Li, et al.European Journal of Medicinal Chemistry|December 29, 2024
Design, synthesis, and biological evaluation of Ponatinib-based N-Phenylpyrimidine-2-amine derivatives as novel fibroblast growth factor receptor 4 (FGFR4) selective inhibitorsLei Han, Yu Yu, Ping Deng, et al.European Journal of Medicinal Chemistry|December 31, 2024
Marine natural product-inspired discovery of novel BRD4 inhibitors with anti-inflammatory activityShuxia Chen, Jichen Yang, Xiangyu Wang, et al.European Journal of Medicinal Chemistry|December 31, 2024
Discovery of the salicylaldehyde-based compound DDO-02267 as a lysine-targeting covalent inhibitor of ALKBH5Wen-Long Fei, Ying-Zhe Wang, Qing-Lan Feng, et al.Pageof 1,614