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Journal of Medicinal Chemistry|September 25, 2018
Discovery of a Potent Thiazolidine Free Fatty Acid Receptor 2 Agonist with Favorable Pharmacokinetic PropertiesAnders Højgaard Hansen, Eugenia Sergeev, Daniele Bolognini, et al.Journal of Medicinal Chemistry|September 26, 2018
Single Amino Acid Substitution in α-Conotoxin TxID Reveals a Specific α3β4 Nicotinic Acetylcholine Receptor AntagonistJinpeng Yu, Xiaopeng Zhu, Peta J Harvey, et al.Journal of Medicinal Chemistry|September 7, 2018
Insights into Current Tropomyosin Receptor Kinase (TRK) Inhibitors: Development and Clinical ApplicationWei Yan, Naga Rajiv Lakkaniga, Francesca Carlomagno, et al.Journal of Medicinal Chemistry|September 29, 2018
Synthesis and Antiviral Evaluation of Carbocyclic Nucleoside Analogs of Nucleoside Reverse Transcriptase Translocation Inhibitor MK-8591 (4'-Ethynyl-2-fluoro-2'-deoxyadenosine)François-René Alexandre, Rachid Rahali, Houcine Rahali, et al.Journal of Medicinal Chemistry|October 2, 2018
Alkyl Sulfinates: Radical Precursors Enabling Drug DiscoveryJoel M Smith, Janice A Dixon, Justine N deGruyter, et al.Journal of Medicinal Chemistry|January 1, 1987
Structure-activity relationships of kadsurenone analoguesM M Ponpipom, R L Bugianesi, D R Brooker, et al.Journal of Medicinal Chemistry|August 29, 2018
First SAR Study for Overriding NRAS Mutant Driven Acute Myeloid LeukemiaHanna Cho, Injae Shin, Eunhye Ju, et al.Journal of Medicinal Chemistry|August 29, 2018
Structure-Based Drug Design of Potent Pyrazole Derivatives against Rhinovirus ReplicationLaurène Da Costa, Els Scheers, Antonio Coluccia, et al.Journal of Medicinal Chemistry|October 9, 2018
Nitro-Group-Containing DrugsKunal Nepali, Hsueh-Yun Lee, Jing-Ping LiouJournal of Medicinal Chemistry|April 1, 1987
Molecular structure of the dihydropyridazinone cardiotonic 1,3-dihydro-3,3-dimethyl-5-(1,4,5,6-tetrahydro-6-oxo-pyridazinyl)- 2H-indol-2-one, a potent inhibitor of cyclic AMP phosphodiesteraseD W Robertson, N D Jones, J H Krushinski, et al.Pageof 3,137