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Journal of Medicinal Chemistry|May 19, 2020
Synthesis and Identification of a Novel Lead Targeting Survivin Dimerization for Proteasome-Dependent DegradationRobert Peery, Kwaku Kyei-Baffour, Zizheng Dong, et al.Journal of Medicinal Chemistry|May 19, 2020
Discovery of (1H-Pyrazolo[3,4-c]pyridin-5-yl)sulfonamide Analogues as Hepatitis B Virus Capsid Assembly Modulators by Conformation ConstraintChunting Wang, Yameng Pei, Lin Wang, et al.Journal of Medicinal Chemistry|May 19, 2020
Anti-HIV-Active Nucleoside Triphosphate ProdrugsXiao Jia, Dominique Schols, Chris MeierJournal of Medicinal Chemistry|May 19, 2020
UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 ReceptorsEdith Bartole, Lukas Grätz, Timo Littmann, et al.Journal of Medicinal Chemistry|June 9, 2020
Drug Induced Liver Injury (DILI). Mechanisms and Medicinal Chemistry Avoidance/Mitigation StrategiesBryan H NormanJournal of Medicinal Chemistry|May 23, 2020
Nanobodies Targeting Prostate-Specific Membrane Antigen for the Imaging and Therapy of Prostate CancerLior Rosenfeld, Amiram Sananes, Yuval Zur, et al.Journal of Medicinal Chemistry|May 21, 2020
Colchicine Alkaloids and Synthetic Analogues: Current Progress and PerspectivesIuliia A Gracheva, Ekaterina S Shchegravina, Hans-Günther Schmalz, et al.Journal of Medicinal Chemistry|May 21, 2020
High-Throughput Screening for the Discovery of Enzyme InhibitorsMatthew D LloydJournal of Medicinal Chemistry|May 12, 2020
Structure-Activity Relationship Study Enables the Discovery of a Novel Berberine Analogue as the RXRα Activator to Inhibit Colon CancerBeibei Xu, Xunjin Jiang, Jing Xiong, et al.Journal of Medicinal Chemistry|May 12, 2020
Discovery of DS-1971a, a Potent, Selective NaV1.7 InhibitorTsuyoshi Shinozuka, Hiroyuki Kobayashi, Sayaka Suzuki, et al.Pageof 3,134