Yuki Tachibana

8PUBLICATIONS
16CO-AUTHORS
Nanoelectromechanical systemsBiologically active moleculesProteins and peptidesCheminformatics and quantitative structure-activity relationshipsMolecular targets
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Publications (8)

|Apr 15, 2026
Structure-Based Drug Discovery of Non-SAM-Mimetic Bisubstrate Inhibitors against Nicotinamide N‑Methyltransferase.

Shuhei Yoshida, Noriyasu Kondo, Shota Uehara

|Jul 05, 2025
Discovery of the Clinical Candidate S-892216: A Second-Generation of SARS-CoV-2 3CL Protease Inhibitor for Treating COVID-19.

Yuto Unoh, Keiichiro Hirai, Shota Uehara

|Nov 17, 2023
Peptide-to-Small Molecule: Discovery of Non-Covalent, Active-Site Inhibitors of β-Herpesvirus Proteases.

Shuhei Yoshida, Yusuke Sako, Eiji Nikaido

|Feb 10, 2023
Efficacy comparison of 3CL protease inhibitors ensitrelvir and nirmatrelvir against SARS-CoV-2 in vitro and in vivo.

Takayuki Kuroda, Haruaki Nobori, Keita Fukao

|Aug 01, 2022
Efficacy of ensitrelvir against SARS-CoV-2 in a delayed-treatment mouse model.

Haruaki Nobori, Keita Fukao, Takayuki Kuroda

|Jul 29, 2022
Peptide-to-Small Molecule: A Pharmacophore-Guided Small Molecule Lead Generation Strategy from High-Affinity Macrocyclic Peptides.

Shuhei Yoshida, Shota Uehara, Noriyasu Kondo

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