Harrie J M Gijsen
14PUBLICATIONS
28CO-AUTHORS
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Publications (14)
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|Feb 17, 2025
Design, Synthesis, and Characterization of GluN2A Negative Allosteric Modulators Suitable for In Vivo Exploration.François P Bischoff, Sven Van Brandt, Marcel Viellevoye
|Feb 11, 2025
Discovery of Potent and Brain-Penetrant Bicyclic NLRP3 Inhibitors with Peripheral and Central In Vivo Activity.Oscar Mammoliti, Rodrigo Carbajo, Laura Perez-Benito
|Jun 05, 2023
European Medicinal Chemistry Leaders in Industry (EMCL) - On the Status and Future of Medicinal Chemistry Research in Europe.Amjad Ali, Marcus Bauser, Sophie Bertrand
|Jan 21, 2022
A Brain-Penetrant and Bioavailable Pyrazolopiperazine BACE1 Inhibitor Elicits Sustained Reduction of Amyloid β In Vivo.Aldo Peschiulli, Daniel Oehlrich, Michiel Van Gool
|Sep 23, 2021
Discovery of Extremely Selective Fused Pyridine-Derived β-Site Amyloid Precursor Protein-Cleaving Enzyme (BACE1) Inhibitors with High In Vivo Efficacy through 10s Loop Interactions.Tatsuhiko Ueno, Eriko Matsuoka, Naoya Asada
|Sep 23, 2021
JNJ-67569762, A 2-Aminotetrahydropyridine-Based Selective BACE1 Inhibitor Targeting the S3 Pocket: From Discovery to Clinical Candidate.Frederik J R Rombouts, Ken-Ichi Kusakabe, Richard Alexander
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Frequent Collaborators
8 joint publications
Kenichi Kusakabe
6 joint publications
Frederik J R Rombouts
4 joint publications
Daniel Oehlrich
3 joint publications
Andrés A Trabanco
1 joint publications
Christoph Boss
1 joint publications
Adrian Hall
1 joint publications
Ruth A Steele
1 joint publications
Ingo V Hartung
1 joint publications
Gilbert Lassalle
1 joint publications
Leena Otsomaa
