Anuradha Gupta
16PUBLICATIONS
57CO-AUTHORS

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Publications (16)
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|Mar 30, 2026
From Flat to 3D: Replacing Phenyl Rings with Saturated Bridged Bicyclic Mimetics to Mitigate Bioactivation and Optimize ADME Properties and Oral Bioavailability in Reverse Amide Orientation.Murugaiah A M Subbaiah, Shruti Surendran, Gaurav Saini
|Dec 03, 2025
Desymmetrization of meso-Anhydride Enabled Enantioselective Synthesis of (-)-7-(Bromomethylene)-3-amidobicyclo[2.2.1]heptane-2-carboxamide, a Scaffold for Divergent Drug Discovery Synthesis.Jianqing Li, Subramaniam Krishnananthan, Daniel Smith
|Oct 01, 2025
Beyond Bioisosteres: Impact of Replacing a Benzene Ring with sp3-Rich Three-Dimensional Saturated Bridged Bicyclic Match Pairs on Biotransformation, Metabolic Stability, and Other ADME Profiles.Shruti Surendran, Sivashankaran Raju, Naveen Kalyani
|May 24, 2025
Discovery and Characterization of a First-in-Class LIV1-TLR7/8 Immunomodulatory Conjugate with Robust Myeloid Activation and Antitumor Activity.Sayumi Yamazoe, Yam Poudel, Emanuela Sega
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Frequent Collaborators
9 joint publications
Vetrichelvan Muthalagu
5 joint publications
James Kempson
3 joint publications
T G Murali Dhar
3 joint publications
Jianqing Li
3 joint publications
Murugaiah A M Subbaiah
3 joint publications
Arvind Mathur
2 joint publications
E Scott Priestley
2 joint publications
Percy H Carter
2 joint publications
Liping Zhang
2 joint publications
Martins S Oderinde