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Updated: Sep 29, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors

James C Sutton1, Scott A Bolton, Karen S Hartl

  • 1The Bristol-Myers Squibb Pharmaceutical Research Institute, PO Box 4000, Princeton, NJ 08543-4000, USA. james.sutton@bms.com

Bioorganic & Medicinal Chemistry Letters
|October 10, 2002
PubMed

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