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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Slow antagonist dissociation and long-lasting in vivo receptor protection

Georges Vauquelin1, Isabelle Van Liefde

  • 1Department of Molecular and Biochemical Pharmacology, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium. gvauquel@vub.ac.be

Trends in Pharmacological Sciences
|June 13, 2006
PubMed

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