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Generation of neutralization-resistant HIV-1 in vitro due to amino acid interchanges of third hypervariable env

T Masuda1, S Matsushita, M J Kuroda

  • 1Department of Biodefence and Medical Virology, Kumamoto University Medical School, Japan.

Insights

HIV-1 variants resistant to a specific antibody targeting the V3 domain of gp120 were developed. Mutations in the V3 region altered viral antigenicity and antibody binding, particularly a key conserved sequence.

Area of Science:

  • Virology
  • Immunology
  • Molecular Biology

Background:

  • Human Immunodeficiency Virus type 1 (HIV-1) envelope glycoprotein gp120 contains the V3 domain, a critical target for neutralizing antibodies.
  • Development of drug resistance is a major challenge in HIV-1 therapy, necessitating understanding of viral evolution under selective pressure.

Purpose of the Study:

  • To investigate the emergence and characteristics of HIV-1 antigenic mutants resistant to a specific neutralizing monoclonal antibody (mAb) targeting the V3 domain.
  • To analyze the genomic and antigenic changes associated with antibody escape.

Main Methods:

  • Isolation of HIV-1 antigenic mutants by passaging plaque-cloned viruses in the presence of mAb 0.5 beta.
  • Nucleotide sequencing to identify genomic variations in isolated mutants.
  • Radioimmunoprecipitation and synthetic peptide analysis to assess binding affinity and antigenic changes.

Main Results:

  • Antigenic HIV-1 mutants resistant to mAb 0.5 beta were successfully isolated.
  • Nucleotide sequencing revealed base substitutions within the V3 domain of resistant mutants, affecting the mAb 0.5 beta binding site.
  • A specific mutation (Pro320 to Gln) in a conserved V3 region significantly reduced binding affinity to mAb 0.5 beta.
  • Other observed mutations did not impact binding affinity in radioimmunoprecipitation assays.
  • Frequent nucleic acid substitutions in the V3 domain occurred even without the selective pressure of mAb 0.5 beta in an in vitro system.

Conclusions:

  • The V3 domain of HIV-1 gp120 is a key target for antibody-mediated neutralization, and mutations within this region can lead to the emergence of resistant variants.
  • Specific amino acid substitutions, particularly in conserved regions like Gly-Pro-Gly-Arg, can significantly alter viral antigenicity and reduce antibody binding affinity.
  • Understanding these escape mechanisms is crucial for developing effective HIV-1 vaccines and therapies.

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