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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Second generation catalytic asymmetric synthesis of Tamiflu: allylic substitution route

Tsuyoshi Mita1, Nobuhisa Fukuda, Francesc X Roca

  • 1Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.

Organic Letters
|January 16, 2007
PubMed

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