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Efficient synthesis and evaluation of bimodal ligand NETA

Hyun-Soon Chong1, Hyun A Song, Noah Birch

  • 1Chemistry Division, Biological, Chemical, and Physical Sciences Department, Illinois Institute of Technology, 3101 S. Dearborn Street, LS 182, Chicago, IL 60616, USA. chong@iit.edu

Bioorganic & Medicinal Chemistry Letters
|May 1, 2008
PubMed
Summary

A novel bimodal ligand, NETA, was synthesized for antibody-targeted radiation therapy. NETA shows promise as a chelator for bismuth and lutetium radioisotopes in cancer treatment.

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