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Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay
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Published on: February 9, 2021

The impact of aromatic ring count on compound developability--are too many aromatic rings a liability in drug design?

Timothy J Ritchie1, Simon J F Macdonald

  • 1Respiratory CEDD, GlaxoSmithKline Research Medicines Centre, Gunnels Wood Road, Stevenage SG1 2NY, UK.

Drug Discovery Today
|September 5, 2009
PubMed

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