[Synthesis and biological activity of 2-dialkylaminoalkoxybenzylidene-benzo-(b)-cyclanones]

¹Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie de Paris-Sud, Châtenay-Malabry.

|January 1, 1990

Abstract:

The synthesis and the study of the cardiovascular and antiallergic properties of 2-(4-dialkylaminoalkoxybenzylidene)-benzo-[b]-1-cyclanones analogues to benzarone and amiodarone were performed. They showed the influence of the length of the basic dialkylaminoalkoxy group and that of a methoxy substitutant of the tetralone on the studied activities.

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Abstract:

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