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Enzyme inhibitor discovery by activity-based protein profiling

Micah J Niphakis1, Benjamin F Cravatt

  • 1The Skaggs Institute for Chemical Biology and the Department of Chemical Physiology, The Scripps Research Institute, La Jolla, California 92037;

Annual Review of Biochemistry
|June 7, 2014
PubMed

Keywords:
activity-based protein profilingchemical proteomicsenzymeinhibitortarget engagement

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